SCHEMBL5889156

SCHEMBL5889156

C[Si](C)(c1ccccc1)C1C=CCCC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
CYP2C19 P33261 1/20 0.35
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889119 0.95 CYP2C19 (0.34) ALDH1A1HPGDAPOBEC3GCYP2C19
SCHEMBL5889273 0.93 NR1H2 (0.33) ALDH1A1HPGDAPOBEC3GCYP2C19
SCHEMBL5889275 0.93 NR1H2 (0.33) ALDH1A1HPGDAPOBEC3GCYP2C19
SCHEMBL5889253 0.89 CYP2C19 (0.37) CYP2C19ESR1ESR2
SCHEMBL19622284 0.77 CES2 (0.32) ALDH1A1HPGD
SCHEMBL6290380 0.73
SCHEMBL23700979 0.68
SCHEMBL2622738 0.68 NR1H2 (0.54) ALDH1A1HPGDESR1ESR2
SCHEMBL5011624 0.68
SCHEMBL10623191 0.68 ALDH1A1 (0.34) ALDH1A1HPGDAPOBEC3G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060194827-A1 5-Cycloalkenyl 5H-chromeno[3,4-f]quinoline derivatives as selective progesterone receptor modulator compounds LIGAND PHARMACEUTICALS, INCORPORATED 2006-08-31 US disclosed
US-7071205-B2 5-cycloalkenyl 5H-chromeno[3,4-f]quinoline derivatives as selective progesterone receptor modulator compounds LIGAND PHARMACEUTICALS INCORPORATED (US) 2006-07-04 US disclosed
EP-1551845-A1 5-CYCLOALKENYL 5 i H /i -CHROMENO 3,4-F QUINOLINE DERIV ATIVES AS SELECTIVE PROGESTERONE RECEPTOR MODULATOR COMPOUNDS LIGAND PHARMACEUTICALS, INC. (US) 2005-07-13 EP disclosed
US-20040152718-A1 5-cycloalkenyl 5H-chromeno[3,4-f]quinoline derivatives as selective progesterone receptor modulator compounds CITIBANK, N.A., AS ADMINISTRATIVE AGENT 2004-08-05 US disclosed
WO-2004033460-A1 5-CYCLOALKENYL 5H-CHROMENO[3,4-F]QUINOLINE DERIVATIVES AS SELECTIVE PROGESTERONE RECEPTOR MODULATOR COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2004-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060194827-A1 5-Cycloalkenyl 5H-chromeno[3,4-f]quinoline derivatives as selective progesterone receptor modulator compounds PGR, GPER1, FSHR ALDH1A1 3556/4885HPGD 474/4885APOBEC3G 4428/4885
US-20040152718-A1 5-cycloalkenyl 5H-chromeno[3,4-f]quinoline derivatives as selective progesterone receptor modulator compounds PGR, GPER1, PGRMC2 ALDH1A1 2500/4885HPGD 551/4885APOBEC3G 4087/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.