SCHEMBL5897906

SCHEMBL5897906

CCCCCc1nc(C)c[nH]1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43
GPR84 Q9NQS5 5/20 0.41
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL83498 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL27699982 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL27680704 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL535754 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL905200 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL24880067 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL9956114 0.98 ALDH1A1 (0.46) ALDH1A1PKMHPGDGPR84KCNH2
Hydrochloric Acid SCHEMBL28365190 0.96 ALDH1A1 (0.44) ALDH1A1PKMHPGDGPR84KCNH2
SCHEMBL9482122 0.96 ALDH1A1 (0.44) ALDH1A1PKMHPGDGPR84KCNH2
Water SCHEMBL28794479 0.96 ALDH1A1 (0.44) ALDH1A1PKMHPGDGPR84KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111315745-B Triazolo-aza derivatives 豪夫迈·罗氏有限公司 2023-07-14 CN disclosed
CN-101182310-B Method for preparing biphenyl substituted pyrimidine compounds UNIV EAST CHINA SCIENCE & TECH 2010-04-14 CN disclosed
CN-101182310-A Method for preparing biphenyl substituted pyrimidine compounds UNIV EAST CHINA SCIENCE & TECH (CN) 2008-05-21 CN disclosed
US-7030144-B2 Substituted imidazole derivatives: GABAA receptor ligands NEUROGEN CORPORATION (US) 2006-04-18 US disclosed
EP-1499608-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES: GABA A RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2005-01-26 EP disclosed
US-20040002608-A1 Substituted imidazole derivatives: GABAA receptor ligands NEUROGEN CORPORATION 2004-01-01 US disclosed
WO-2003093263-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES: GABAA RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2003-11-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040002608-A1 Substituted imidazole derivatives: GABAA receptor ligands GABRA1, GABRA3, GABRA2 ALDH1A1 719/4885PKM 1540/4885HPGD 2526/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.