Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL5898930

CCO.ClCCl.O=C(O)C(F)(F)F

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

MMP1MMP13MMP7MMP8polrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Trifluoroacetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FAAH O00519 8/20 0.36
FUCA1 P04066 1/20 0.35
CES1 P23141 5/20 0.34
CES2 O00748 3/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TSHR P16473 4/20 0.33
ALDH1A1 P00352 3/20 0.33
FFAR3 O14843 1/20 0.33
TP53 P04637 1/20 0.33
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3794549 0.91 FAAH (0.40) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL30324569 0.91 FAAH (0.40) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL281599 0.91 FAAH (0.40) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL5382443 0.91 FAAH (0.50) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL4872786 0.88 TSHR (0.37) FAAHCES1CES2MEN1CYP1A2
Trifluoroacetic Acid SCHEMBL21924385 0.88 FAAH (0.39) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL27627328 0.88 FAAH (0.39) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL6909668 0.88 FAAH (0.39) FAAHFUCA1CES1CES2MEN1
Trifluoroacetic Acid SCHEMBL6950012 0.88 FAAH (0.39) FAAHCES1CES2MEN1CYP1A2
Trifluoroacetic Acid SCHEMBL27681955 0.88 FAAH (0.39) FAAHFUCA1CES1CES2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2944637-B1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2020-02-19 EP disclosed
CN-104903320-B Nitrogen-containing heterocycle compound or its salt 富士胶片株式会社 2018-11-13 CN disclosed
US-9783536-B2 Nitrogen-containing heterocyclic compound or salt thereof FUJIFILM CORPORATION (JP) 2017-10-10 US disclosed
CN-104535673-B A kind of method of HPLC separation determination rosuvastain calcium enantiomter SUNSHINE LAKE PHARMA CO.,LTD. (CN) 2016-04-20 CN disclosed
EP-2944637-A1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM Corporation (JP) 2015-11-18 EP disclosed
US-20150322063-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND OR SALT THEREOF FUJIFILM CORPORATION (JP) 2015-11-12 US disclosed
CN-104903320-A Nitrogen-containing heterocylic compound or salt thereof FUJIFILM CORP 2015-09-09 CN disclosed
CN-104535673-A Method for separating and measuring enantiomer of rosuvastatin calcium via HPLC GUANGDONG HEC PHARMACEUTICAL 2015-04-22 CN disclosed
US-20060058346-A1 Novel enantiomers of etrahydroisoquinoline derivatives and theirpharmaceutically acceptable salts, their preparations and pharmaceutical compositions YUN-CHOI HYE-SOOK 2006-03-16 US disclosed
EP-0671975-B2 CHIRAL ADSORBENTS AND PREPARATION THEREOF AS WELL AS COMPOUNDS ON WHICH THE ADSORBENTS ARE BASED AND PREPARATION OF THESE COMPOUNDS EKA CHEMICALS AB (SE) 2002-07-03 EP disclosed
US-6333426-B1 CHIRAL STATIONARY PHASES BASED ON NETWORK POLYMERS OF TARTARIC ACID DERIVATIVES EXHIBIT GENERAL ENANTIOSELECTIVITY FOR MOST TYPES OF PHARMACEUTICAL SUBSTANCES EKA NOBEL AB (SE) 2001-12-25 US disclosed
US-6277782-B1 POLYMER BONDED TO CARRIER EKA NOBEL AB (SE) 2001-08-21 US disclosed
EP-0671975-B1 CHIRAL ADSORBENTS AND PREPARATION THEREOF AS WELL AS COMPOUNDS ON WHICH THE ADSORBENTS ARE BASED AND PREPARATION OF THESE COMPOUNDS EKA CHEMICALS AB (SE) 1998-07-22 EP disclosed
EP-0671975-A1 CHIRAL ADSORBENTS AND PREPARATION THEREOF AS WELL AS COMPOUNDS ON WHICH THE ADSORBENTS ARE BASED AND PREPARATION OF THESE COMPOUNDS Eka Chemicals AB (SE) 1995-09-20 EP disclosed
WO-1994012275-A1 CHIRAL ADSORBENTS AND PREPARATION THEREOF AS WELL AS COMPOUNDS ON WHICH THE ADSORBENTS ARE BASED AND PREPARATION OF THESE COMPOUNDS EKA NOBEL AB (SE) 1994-06-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060058346-A1 Novel enantiomers of etrahydroisoquinoline derivatives and theirpharmaceutically acceptable salts, their preparations and pharmaceutical compositions TBXA2R, NOS2, TBXAS1 FAAH 1250/4885FUCA1 4677/4885CES1 960/4885
US-20150322063-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND OR SALT THEREOF NPM1, NAP1L1, REN FAAH 2685/4885FUCA1 4043/4885CES1 1795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.