SCHEMBL5917

SCHEMBL5917

O=Cc1ccc(-c2nnn[nH]2)cc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.35
HSD17B10 Q99714 1/20 0.35
ALDH5A1 P51649 1/20 0.35
ABAT P80404 1/20 0.35
BRD4 O60885 1/20 0.35
KCNJ1 P48048 2/20 0.34
DRD1 P21728 2/20 0.34
ALDH1A1 P00352 5/20 0.33
KDM4E B2RXH2 2/20 0.32
TYR P14679 1/20 0.32
CYP2A13 Q16696 1/20 0.32
KIF11 P52732 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1561472 0.83 DRD1 (0.42) CYP2A6BRD4KCNJ1DRD1ALDH1A1
SCHEMBL2028396 0.83 ADH5 (0.32)
SCHEMBL1562532 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
SCHEMBL1562221 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
Lithium SCHEMBL1562536 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
SCHEMBL1561381 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
SCHEMBL1561389 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
Potassium SCHEMBL1561386 0.82 DRD1 (0.41) CYP2A6DRD1ALDH1A1
SCHEMBL13411813 0.81 ADH5 (0.36)
SCHEMBL5950535 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 84 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116283701-B Compounds having the structure 4- (substituted aminomethyl) -5-neopentyl-N-substituted pyrrolidine-2-carboxamide 中国科学院上海药物研究所 2025-04-22 CN disclosed
US-12173018-B2 Penicillin-binding protein inhibitors VenatoRx Pharmaceuticals, Inc. (US) 2024-12-24 US disclosed
CN-117120416-A Small molecule compound with substituted phenyl spiro [ indoline-3, 3' -pyrrolidine ] structure 中国科学院上海药物研究所 2023-11-24 CN disclosed
CN-116283701-A Compounds having the structure 4- (substituted aminomethyl) -5-neopentyl-N-substituted pyrrolidine-2-carboxamide 中国科学院上海药物研究所 2023-06-23 CN disclosed
US-11613535-B2 Compounds for MYC inhibition THE SCRIPPS RESEARCH INSTITUTE (US) 2023-03-28 US disclosed
EP-3820847-B1 IMPROVED COMPOUNDS FOR MYC INHIBITION SCRIPPS RESEARCH INST (US) 2022-12-14 EP disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-115215872-A Small molecule compound with substituted phenyl spiro [ indoline-3, 3' -pyrrolidine ] structure 中国科学院上海药物研究所 2022-10-21 CN disclosed
WO-2022218379-A1 SMALL-MOLECULE COMPOUND HAVING SUBSTITUTED PHENYL SPIRO[INDOLINE-3,3'-PYRROLIDINE] STRUCTURE 中国科学院上海药物研究所 2022-10-20 WO disclosed
US-20220227765-A1 PYRIDO-INDOLE ANALOGUES AS GPX4 INHIBITORS ADRENAS THERAPEUTICS INC. 2022-07-21 US disclosed
US-6110946-A AN ENZYME INHIBITORS OF RETROVIRAL ASPARTATE PROTEASE FOR THE TREATMENT OF AIDS NOVARTIS FINANCE CORPORATION (US) 2000-08-29 US disclosed
EP-0983251-A1 ANTI-INFLAMMATORY PIPERAZINYL-BENZYL-TETRAZOLE DERIVATIVES AND INTERMEDIATES THEREOF Pfizer Limited (GB) 2000-03-08 EP disclosed
EP-0929553-A1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Novartis AG (CH) 1999-07-21 EP disclosed
EP-0900210-A1 ANTIVIRALLY ACTIVE HETEROCYCLIC AZAHEXANE DERIVATIVES Novartis AG (CH) 1999-03-10 EP disclosed
US-5849911-A Antivirally active heterocyclic azahexane derivatives NOVARTIS FINANCE CORPORATION (US) 1998-12-15 US disclosed
WO-1998052929-A1 ANTI-INFLAMMATORY PIPERAZINYL-BENZYL-TETRAZOLE DERIVATIVES AND INTERMEDIATES THEREOF PFIZER LIMITED (GB) 1998-11-26 WO disclosed
WO-1998014450-A1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 1998-04-09 WO disclosed
WO-1997040029-A1 ANTIVIRALLY ACTIVE HETEROCYCLIC AZAHEXANE DERIVATIVES NOVARTIS AG (CH) 1997-10-30 WO disclosed
US-RE32196-E PROPHYLACTIC CHEMOTHERAPY OF ALLERGIC CONDITIONS LILLY INDUSTRIES LIMITED (GB) 1986-07-01 US disclosed
US-4259340-A PROPHYLACTIC CHEMOTHERAPY OF ALLERGIC CONDITIONS SUCH AS ASTHMA LILLY INDUSTRIES LIMITED (GB) 1981-03-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11613535-B2 Compounds for MYC inhibition MYC, MYCBP, MYCBP2 CYP2A6 3559/4885HSD17B10 4157/4885ALDH5A1 3715/4885
US-12173018-B2 Penicillin-binding protein inhibitors PEPD, BPGM, EBPL CYP2A6 2454/4885HSD17B10 2285/4885ALDH5A1 3327/4885
US-20220227765-A1 PYRIDO-INDOLE ANALOGUES AS GPX4 INHIBITORS GPX4, GPX1, AIFM2 CYP2A6 1942/4885HSD17B10 1195/4885ALDH5A1 139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.