SCHEMBL592290

SCHEMBL592290

COc1cccc(-c2nc3ccccc3o2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.72
HPGD P15428 7/20 0.72
NPC1 O15118 6/20 0.72
RAB9A P51151 6/20 0.72
SMN1; SMN2 Q16637 6/20 0.72
HSD17B10 Q99714 6/20 0.72
KDM4E B2RXH2 5/20 0.72
TP53 P04637 4/20 0.72
NFKB1 P19838 3/20 0.72
NFKB2 Q00653 3/20 0.72
RELA Q04206 3/20 0.72
TDP1 Q9NUW8 2/20 0.72
L3MBTL1 Q9Y468 2/20 0.72
GLA P06280 1/20 0.72
KMT2A Q03164 2/20 0.67
F2 P00734 1/20 0.67
CASP3 P42574 2/20 0.63
LMNA P02545 1/20 0.63
P2RY14 Q15391 2/20 0.61
PTPN2 P17706 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052772 0.87 NPC1 (0.69) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL12639231 0.86 RAB9A (0.74) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL4051577 0.86 SMN1; SMN2 (0.74) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL4059683 0.86 NPC1 (0.65) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL4052671 0.84 NPC1 (0.62) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL376001 0.84 ALDH1A1 (0.64) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL4054520 0.83 SMN1; SMN2 (0.74) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL4053543 0.83 NPC1 (0.65) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL1199992 0.83 PTPN2 (0.68) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL27520950 0.82 ALDH1A1 (0.64) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250381221-A1 Compositions and Methods for Treating Cancer IN8BIO INC (US) 2025-12-18 US disclosed
US-20250161247-A1 METHOD FOR TREATING BREAST CANCERS AND PARP RESISTANT BREAST CANCERS LANTERN PHARMA INC. (US) 2025-05-22 US disclosed
EP-4554683-A2 METHOD FOR TREATING BREAST CANCERS AND PARP RESISTANT BREAST CANCERS Lantern Pharma Inc. (US) 2025-05-21 EP disclosed
US-20240299322-A1 TREATING CANCERS WITH COMBINATIONS OF PARP INHIBITOR AND ACYLFULVENES LANTERN PHARMA INC. (US) 2024-09-12 US disclosed
US-20240245643-A1 DNA Damage Repair Inhibitors for Treatment of Cancer THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2024-07-25 US disclosed
WO-2024016014-A2 METHOD FOR TREATING BREAST CANCERS AND PARP RESISTANT BREAST CANCERS LANTERN PHARMA INC. (US) 2024-01-18 WO disclosed
US-20230255906-A1 Targeting Serpin B9 in Cancer THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2023-08-17 US disclosed
US-20220339179-A1 TREATMENT OF HR DEFICIENT CANCER THE FRANCIS CRICK INSTITUTE LIMITED (GB) 2022-10-27 US disclosed
EP-4028009-A1 TREATMENT OF HR DEFICIENT CANCER The Francis Crick Institute Limited (GB) 2022-07-20 EP disclosed
US-11162095-B2 Use of a combination of Dbait molecule and PARP inhibitors to treat cancer INSTITUT CURIE (FR) 2021-11-02 US disclosed
EP-2167086-A1 COMBINATION OF CHK AND PARP INHIBITORS FOR THE TREATMENT OF CANCERS AstraZeneca AB (SE) 2010-03-31 EP disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
WO-2008146035-A1 COMBINATION OF CHK AND PARP INHIBITORS FOR THE TREATMENT OF CANCERS ASTRAZENECA AB (SE) 2008-12-04 WO disclosed
WO-2008020180-A2 METHODS OF INCREASING THE SENSITIVITY OF CANCER CELLS TO DNA DAMAGE KUDOS PHARMACEUTICALS LIMITED (GB) 2008-02-21 WO disclosed
EP-1684736-A1 DNA DAMAGE REPAIR INHIBITORS FOR TREATMENT OF CANCER Kudos Pharmaceuticals Limited (GB) 2006-08-02 EP disclosed
US-20060142231-A1 DNA damage repair inhibitors for treatment of cancer KUDOS PHARMACEUTICALS LIMITED (GB) 2006-06-29 US disclosed
US-20050227919-A1 DNA damage repair inhibitors for the treatment of cancer KUDOS PHARMACEUTICALS LIMITED 2005-10-13 US disclosed
WO-2005053662-A1 DNA DAMAGE REPAIR INHIBITORS FOR TREATMENT OF CANCER KUDOS PHARMACEUTICALS LIMITED (GB) 2005-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250161247-A1 METHOD FOR TREATING BREAST CANCERS AND PARP RESISTANT BREAST CANCERS PARP1, PARP2, PARP3 ALDH1A1 1781/4885HPGD 1833/4885NPC1 4253/4885
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION DBH, DDT, CYCS ALDH1A1 117/4885HPGD 1702/4885NPC1 1565/4885
US-11162095-B2 Use of a combination of Dbait molecule and PARP inhibitors to treat cancer PARP10, PARP1, PARP3 ALDH1A1 349/4885HPGD 1350/4885NPC1 3786/4885
US-20240299322-A1 TREATING CANCERS WITH COMBINATIONS OF PARP INHIBITOR AND ACYLFULVENES PARP1, PARP2, PARP11 ALDH1A1 1466/4885HPGD 1722/4885NPC1 3852/4885
US-20240245643-A1 DNA Damage Repair Inhibitors for Treatment of Cancer PARP2, MRE11, PARP1 ALDH1A1 747/4885HPGD 325/4885NPC1 4490/4885
US-20060142231-A1 DNA damage repair inhibitors for treatment of cancer MRE11, PARP2, ERCC4 ALDH1A1 744/4885HPGD 359/4885NPC1 4486/4885
US-20230255906-A1 Targeting Serpin B9 in Cancer SERPINB10, SERPINB8, SERPINE1 ALDH1A1 3233/4885HPGD 1255/4885NPC1 1048/4885
US-20050227919-A1 DNA damage repair inhibitors for the treatment of cancer MRE11, ERCC4, PARP2 ALDH1A1 729/4885HPGD 313/4885NPC1 4509/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.