SCHEMBL5952745

SCHEMBL5952745

C[Sn](C)(C)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
ALDH1A1 P00352 4/20 0.45
ALOX15 P16050 2/20 0.38
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
CA2 P00918 3/20 0.33
NOS1 P29475 2/20 0.33
CA1 P00915 2/20 0.33
TSHR P16473 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
TAAR1 Q96RJ0 3/20 0.32
HSP90AA1 P07900 1/20 0.31
TLR9 Q9NR96 1/20 0.31
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1593230 0.83
SCHEMBL31198155 0.73 CYP2A6 (0.57) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL8585311 0.73 ALDH1A1 (0.32) ALDH1A1TDP1
SCHEMBL904638 0.71 ACHE (0.53) CYP2A6ALDH1A1TDP1CA2CA1
SCHEMBL18508 0.71
SCHEMBL7384302 0.69 TRPA1 (0.43) ALDH1A1TSHRCES2CES1
SCHEMBL2392186 0.69 LMNA (0.50) CYP2A6ALDH1A1MAPK1HDAC8TSHR
SCHEMBL5951790 0.69 CYP3A4 (0.50) ALDH1A1ALOX15MAPK1CA2CA1
SCHEMBL979413 0.69 ACHE (0.45) CA2NOS1CA1CES2CES1
SCHEMBL5951383 0.69 MEN1 (0.50) ALDH1A1ALOX15MAPK1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed
US-5541169-A FUNGICIDES KOWA COMPANY, LTD. (JP) 1996-07-30 US disclosed
EP-0632021-A1 AZOXY COMPOUND KOWA CO. LTD. (JP) 1995-01-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A CYP2A6 64/4885ALDH1A1 317/4885ALOX15 3737/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 CYP2A6 78/4885ALDH1A1 198/4885ALOX15 3758/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.