SCHEMBL5956691

SCHEMBL5956691

Cc1ccnc(-c2ccc(Br)cc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.61
CCR5 P51681 1/20 0.61
CCR8 P51685 1/20 0.61
CYP2A6 P11509 1/20 0.53
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
KDM4E B2RXH2 4/20 0.50
PIK3CA P42336 1/20 0.50
PIK3CG P48736 1/20 0.50
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
APP P05067 1/20 0.46
PAX8 Q06710 1/20 0.46
UHRF1 Q96T88 1/20 0.45
METAP2 P50579 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31695263 0.89 CCR1 (0.76) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL27344644 0.89 CCR1 (0.76) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL29463685 0.85 CCR1 (0.70) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL6807225 0.85 CCR1 (0.70) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL28660538 0.83 ALDH1A1 (0.46) CCR1CCR5CCR8NPC1RAB9A
SCHEMBL28630968 0.83 ALDH1A1 (0.46) CCR1CCR5CCR8NPC1RAB9A
SCHEMBL16210551 0.81 MEN1 (0.47) NPC1RAB9AKDM4EPIK3CAPIK3CG
SCHEMBL5699981 0.80 KDM1A (0.46) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL2190158 0.80 CYP2A6 (0.62) CCR1CCR5CCR8CYP2A6NPC1
SCHEMBL6183900 0.80 CCR1 (0.61) CCR1CCR5CCR8CYP2A6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108467412-A A kind of green-yellow light phenylpyridine complex of iridium and its preparation method and application 南京邮电大学 2018-08-31 CN claimed
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed
CN-108467412-A A kind of green-yellow light phenylpyridine complex of iridium and its preparation method and application 南京邮电大学 2018-08-31 CN disclosed
US-9478750-B2 Anthracene derivative and organic electroluminescent element using the same JNC CORPORATION (JP) 2016-10-25 US disclosed
CN-103958471-B Anthracene derivant and use its organic electric field luminescence assembly, electron transport material, display device and lighting device 捷恩智株式会社 2016-08-17 CN disclosed
CN-103958471-A Anthracene derivative and organic electroluminescent element using same JNC CORP 2014-07-30 CN disclosed
US-20060004051-A1 Compounds DODIC NERINA 2006-01-05 US disclosed
US-20050245520-A1 2-Phenylpyridin-4-yl derivatives as alk5 inhibitors DODIC NERINA 2005-11-03 US disclosed
EP-1554275-A2 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-20 EP disclosed
WO-2004013134-A2 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245520-A1 2-Phenylpyridin-4-yl derivatives as alk5 inhibitors SMAD2, SMAD3, ALK CCR1 1244/4885CCR5 327/4885CCR8 1108/4885
US-20060004051-A1 Compounds SMAD3, SMAD2, TGFBR1 CCR1 1707/4885CCR5 263/4885CCR8 2319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.