SCHEMBL5969908

SCHEMBL5969908

Cc1cccc(N(Cc2ccc(C(F)(F)F)cc2)C2CCN(C(=O)O)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.43
KCNH2 Q12809 2/20 0.43
DCUN1D1 Q96GG9 4/20 0.42
UBE2M P61081 3/20 0.42
CYP3A4 P08684 1/20 0.41
AR P10275 1/20 0.41
TACR1 P25103 1/20 0.40
MDM2 Q00987 1/20 0.40
PGR P06401 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TEAD1 P28347 1/20 0.40
CETP P11597 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ALDH1A1 P00352 2/20 0.39
AGTR2 P50052 1/20 0.39
USP2 O75604 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5969454 0.89 HSD11B1 (0.44) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL5969537 0.89 CCR5 (0.49) CCR5KCNH2DCUN1D1UBE2MCYP3A4
SCHEMBL4312474 0.88 MEN1 (0.44) CCR5KCNH2DCUN1D1UBE2MCYP3A4
SCHEMBL5969609 0.88 CCR5 (0.47) CCR5KCNH2DCUN1D1UBE2MCYP3A4
SCHEMBL4306650 0.88 MEN1 (0.52) TACR1JAK2
SCHEMBL5969490 0.87 LMNA (0.48) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL5969485 0.85 UBE2M (0.39) CCR5KCNH2DCUN1D1UBE2MTACR1
SCHEMBL5969498 0.85 CHRM1 (0.43) CCR5KCNH2DCUN1D1UBE2MPGR
SCHEMBL5969544 0.83 S1PR1 (0.45) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL5969511 0.83 CETP (0.45) CCR5KCNH2DCUN1D1UBE2MPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556045-B1 4-AMINOPIPERIDINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS UCB SA (BE) 2006-08-02 EP claimed