Pyruvate

Pyruvate

SCHEMBL597153

CC(=O)C(=O)[O-].CC(=O)C(=O)[O-].[Mn+2]

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA4 P22748 3/20 0.91
CA1 P00915 2/20 0.58
TSHR P16473 1/20 0.50
THPO P40225 1/20 0.50
FAHD1 Q6P587 1/20 0.46
LMNA P02545 2/20 0.42
FFAR3 O14843 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
BLM P54132 3/20 0.38
MEN1 O00255 1/20 0.38
LDHA P00338 1/20 0.38
KMT2A Q03164 1/20 0.38
PMP22 Q01453 2/20 0.36
ALOX15 P16050 1/20 0.36
THRB P10828 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyruvate SCHEMBL148220 0.95
Pyruvate SCHEMBL6743471 0.91 CA4 (0.91) CA4CA1TSHRTHPOFAHD1
Pyruvate SCHEMBL7936306 0.91 CA4 (0.91) CA4CA1TSHRTHPOFAHD1
Pyruvate SCHEMBL1331761 0.91
Pyruvate SCHEMBL598199 0.91
Pyruvate SCHEMBL1332703 0.91
Pyruvate SCHEMBL3745552 0.91 CA4 (0.91) CA4CA1TSHRTHPOFAHD1
Pyruvate SCHEMBL18226 0.91
Pyruvate SCHEMBL1332958 0.91
Pyruvate SCHEMBL597752 0.91 CA4 (0.91) CA4CA1TSHRTHPOFAHD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 296 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210393558-A1 METHODS AND COMPOSITIONS FOR PREVENTION AND TREATMENT OF PRESSURE ULCERS TECHNION RES & DEVELOPMENT FOUND LTD (IL) 2021-12-23 US claimed
WO-2021040673-A1 METHODS FOR THE TREATMENT OF CHRONIC HYPOXEMIA AND INHIBITING LUNG FIBROSIS IN PATIENTS WITH PULMONARY FIBROSIS WITH AND WITHOUT COPD MARTIN ALAIN (US) 2021-03-04 WO claimed
EP-3731838-A2 METHODS AND COMPOSITIONS FOR PREVENTION AND TREATMENT OF PRESSURE ULCERS Technion - Research & Development Foundation Ltd (IL) 2020-11-04 EP claimed
CN-104998264-B Methods and compositions for treating mammalian diseases and wounds caused by peroxynitrite overexpression 北方细胞制药公司 2020-09-15 CN claimed
US-20180344621-A1 Methods of Reducing Hair Loss and/or Facilitating Hair Growth and/or Regrowth KENVUE BRANDS LLC 2018-12-06 US claimed
US-20180338936-A1 Methods and Compositions for the Treatment and Prevention of Allergic Rhinitis MARTIN ALAIN (US) 2018-11-29 US claimed
EP-2512418-B1 METHODS OF REDUCING HAIR LOSS AND / OR FACILITATING HAIR GROWTH AND / OR REGROWTH JOHNSON & JOHNSON CONSUMER INC (US) 2017-11-01 EP claimed
US-20170202771-A1 Methods of Reducing Hair Loss and/or Facilitating Hair Growth and/or Regrowth KENVUE BRANDS LLC 2017-07-20 US claimed
US-9675569-B2 Method for treating a pulmonary disease state in mammals by up regulating indigenous in vivo levels of inflammatory agents in mammalian cells CELLULAR SCIENCES, INC. 2017-06-13 US claimed
US-20160022616-A1 Method for Treating a Pulmonary Disease State in Mammals by Up Regulating Indigenous in vivo Levels of Inflammatory Agents in Mammalian Cells CELLULAR SCIENCES, INC. 2016-01-28 US claimed
US-5602183-A DIAPER DERMATITIS; MIXTURE OF ANTIINFLAMMATORY AGENT ANDPYRUVATE COMPOUND, ANTIOXIDANT AND FATTY ACIDS WARNER-LAMBERT COMPANY (US) 1997-02-11 US claimed
WO-1996006640-A9 BIOADHESIVE-WOUND HEALING COMPOSITION 1996-04-11 WO claimed
WO-1996003149-A1 ANTIFUNGAL-WOUND HEALING COMPOSITIONS AND METHODS FOR PREPARING AND USING SAME WARNER-LAMBERT COMPANY (US) 1996-02-08 WO claimed
WO-1995019178-A1 METHODS AND COMPOSITIONS FOR TREATMENT AND DIAGNOSIS OF ALZHEIMER DISEASE AND OTHER DISORDERS RESEARCH FOUNDATION FOR MENTAL HYGIENE, INC. (US) 1995-07-20 WO claimed
EP-0627917-A1 CYTOPROTECTIVE COMPOSITIONS CONTAINING PYRUVATE AND ANTIOXIDANTS WARNER-LAMBERT COMPANY (US) 1994-12-14 EP claimed
EP-0614359-A1 WOUND HEALING COMPOSITIONS CONTAINING A PYRUVATE, AN ANTIOXIDANT AND A MIXTURE OF FATTY ACIDS WARNER-LAMBERT COMPANY (US) 1994-09-14 EP claimed
EP-0573465-A1 THERAPEUTIC COMPOSITIONS TO PROTECT AND RESUSCITATE MAMMALIAN CELLS AND METHODS FOR PREPARING AND USING SAME. WARNER LAMBERT CO (US) 1993-12-15 EP claimed
WO-1993016690-A1 CYTOPROTECTIVE COMPOSITIONS CONTAINING PYRUVATE AND ANTIOXIDANTS WARNER-LAMBERT COMPANY (US) 1993-09-02 WO claimed
WO-1993010776-A1 WOUND HEALING COMPOSITIONS CONTAINING A PYRUVATE, AN ANTIOXIDANT AND A MIXTURE OF FATTY ACIDS WARNER-LAMBERT COMPANY (US) 1993-06-10 WO claimed
WO-1992015292-A1 THERAPEUTIC COMPOSITIONS TO PROTECT AND RESUSCITATE MAMMALIAN CELLS AND METHODS FOR PREPARING AND USING SAME WARNER-LAMBERT COMPANY (US) 1992-09-17 WO claimed