SCHEMBL5971900

SCHEMBL5971900

COCNC(=O)[C@@]12CC[C@@H](C[C@@H](c3ccc(F)cc3)C1)N2C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.39
KCNH2 Q12809 2/20 0.39
SLC6A3 Q01959 10/20 0.38
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
TACR1 P25103 1/20 0.35
SLC18A3 Q16572 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HRH1 P35367 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3422811 1.00 CCR2 (0.39) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL8481404 0.85 OPRK1 (0.42) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL30899722 0.85 OPRK1 (0.42) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL9405511 0.81 DRD2 (0.38) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL9405512 0.81 DRD2 (0.38) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL3422161 0.80 DRD2 (0.38) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL5637165 0.80 DRD2 (0.38) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL3421132 0.80 DRD2 (0.38) CCR2KCNH2SLC6A3SLC6A2SLC6A4
SCHEMBL23924861 0.74 SLC6A3 (0.40) SLC6A3SLC6A2SLC6A4
SCHEMBL3655052 0.73 SLC6A4 (0.41) SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1429811-A4 THEURAPEUTIC TROPANE COMPOUNDS HARVARD COLLEGE (US) 2006-05-17 EP disclosed
EP-1429811-A1 THEURAPEUTIC TROPANE COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2004-06-23 EP disclosed
WO-2003015830-A1 THEURAPEUTIC TROPANE COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2003-02-27 WO disclosed