SCHEMBL5986339

SCHEMBL5986339

CCCCc1ccc(C#Cc2ccc(CN(Cc3ccc(OC(C)=O)cc3)C(=O)c3ccc(O)nc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.41
TP53 P04637 2/20 0.41
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.40
PTPN11 Q06124 1/20 0.38
PTPRO Q16827 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855320 0.89 LPAR1 (0.46) TP53MAPTPOLBPTPN11PTPRO
SCHEMBL13708345 0.87 ACACB (0.40) ACACBTP53MAPTPOLB
SCHEMBL5497713 0.76 THRB (0.46) ACACBPTPN11PTPROTHRB
SCHEMBL5507735 0.76 PTGES (0.54) ACACBPTPN11PTPROTHRB
SCHEMBL2853046 0.74 THRB (0.45) ACACBPTPN11PTPROTHRB
SCHEMBL2858233 0.73 ACACB (0.46) ACACBTHRB
SCHEMBL4055579 0.72 THRB (0.55) ACACBTHRB
SCHEMBL4464485 0.72 STAT3 (0.42) PTPN11PTPROTHRB
SCHEMBL1415501 0.72 THRB (0.61) POLBTHRB
SCHEMBL5501954 0.72 PSMB5 (0.44) ACACBMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-A1 ALKYNYL ARYL CARBOXAMIDES Applied Research Systems ARS Holding N.V. (AN) 2006-05-10 EP disclosed
WO-2005012280-A1 ALKYNYL ARYL CARBOXAMIDES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2005-02-10 WO disclosed