SCHEMBL5990806

SCHEMBL5990806

[CH2]c1ccnc(-c2ccccc2F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.51
TGFBR1 P36897 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
MAPKAPK2 P49137 2/20 0.43
MAPK14 Q16539 2/20 0.43
PLK4 O00444 1/20 0.43
MAPK13 O15264 1/20 0.43
DAPK3 O43293 1/20 0.43
DYRK3 O43781 1/20 0.43
RPS6KA4 O75676 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43
EGFR P00533 1/20 0.43
CDK1 P06493 1/20 0.43
MET P08581 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1938816 0.81 NPC1 (0.51) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL10153369 0.78 NPC1 (0.51) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL4509227 0.78 CCR1 (0.57) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL16488518 0.78 NPC1 (0.51) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL30420906 0.78 ASIC3 (0.56) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL25011838 0.78 ASIC3 (0.56) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL28013790 0.78 NPC1 (0.51) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL28726696 0.75 NPC1 (0.49) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL19817233 0.74 NPC1 (0.60) NPC1TGFBR1L3MBTL1CASP3SENP8
SCHEMBL29857433 0.74 NPC1 (0.60) NPC1TGFBR1L3MBTL1CASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060287378-A1 Novel pyrroles and imidazoles WARNER-LAMBERT COMPANY LLC 2006-12-21 US disclosed
US-20050239857-A1 Novel imidazoles BOLTON GARY L 2005-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060287378-A1 Novel pyrroles and imidazoles PPIP5K2, PPIE, PPOX NPC1 3514/4885TGFBR1 4860/4885L3MBTL1 4821/4885
US-20050239857-A1 Novel imidazoles HMGCR, HMGB2, HMGB3 NPC1 120/4885TGFBR1 3392/4885L3MBTL1 4624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.