SCHEMBL5996017

SCHEMBL5996017

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nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.59
ACE P12821 3/20 0.58
ITGB3 P05106 1/20 0.56
ITGA2B P08514 1/20 0.56
CA2 P00918 1/20 0.56
MME P08473 3/20 0.53
GPR34 Q9UPC5 2/20 0.52
CPA1 P15085 2/20 0.51
ACE2 Q9BYF1 2/20 0.51
FOLH1 Q04609 2/20 0.50
POLB P06746 1/20 0.50
GNPAT O15228 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
PAM P19021 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL504108 1.00 ALDH1A1 (0.61) ALDH1A1LMNAACEITGB3ITGA2B
SCHEMBL27547070 1.00 ALDH1A1 (0.61) ALDH1A1LMNAACEITGB3ITGA2B
Valine SCHEMBL7689739 0.89 ALDH1A1 (0.51) ALDH1A1LMNAACEITGB3ITGA2B
SCHEMBL5995731 0.89 MME (0.63) ALDH1A1LMNAACEMMECPA1
SCHEMBL31688037 0.87 MME (0.52) ALDH1A1LMNAACEITGB3ITGA2B
Acetyl Tyrosine SCHEMBL8977600 0.85 FOLH1 (0.66) LMNAACEITGB3ITGA2BCA2
SCHEMBL5061764 0.85 LMNA (0.61) LMNAACEITGB3ITGA2BMME
Acetyl Tyrosine SCHEMBL8977601 0.85 FOLH1 (0.66) LMNAACEITGB3ITGA2BCA2
SCHEMBL14031836 0.85 LMNA (0.61) LMNAACEITGB3ITGA2BMME
SCHEMBL11122115 0.85 LMNA (0.61) LMNAACEITGB3ITGA2BMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377589-B1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS PHARMACIA ITALIA SPA (IT) 2005-09-07 EP claimed
WO-2002068586-A2 HIV/FIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2002-09-06 WO claimed
EP-4661890-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS Purdue Research Foundation (US) 2025-12-17 EP disclosed
WO-2024167565-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS PURDUE RESEARCH FOUNDATION (US) 2024-08-15 WO disclosed
US-20230257388-A1 GRANZYME B DIRECTED IMAGING AND THERAPY CYTOSITE BIOPHARMA INC. (US) 2023-08-17 US disclosed
US-11667645-B2 Granzyme B directed imaging and therapy CYTOSITE BIOPHARMA INC. (US) 2023-06-06 US disclosed
WO-2021119554-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY KUMQUAT BIOSCIENCES INC. (US) 2021-06-17 WO disclosed
CN-112261939-A Granzyme B directed imaging and therapy 塞托赛特生物制药股份有限公司 2021-01-22 CN disclosed
EP-3752145-A1 GRANZYME B DIRECTED IMAGING AND THERAPY Cytosite Biopharma Inc. (US) 2020-12-23 EP disclosed
US-20200369673-A1 GRANZYME B DIRECTED IMAGING AND THERAPY CYTOSITE BIOPHARMA INC. 2020-11-26 US disclosed
EP-3634498-A1 LINKED AND OTHER PH-TRIGGERED COMPOUNDS Rhode Island Council on Postsecondary Education (US) 2020-04-15 EP disclosed
CN-1155612-C Endothelin antagon 中国人民解放军军事医学科学院毒物药 2004-06-30 CN disclosed
EP-1365023-A1 DNA ENCODING NOVEL D-AMINOACYLASE AND PROCESS FOR PRODUCING D-AMINO ACID BY USING THE SAME Mitsui Chemicals, Inc. (JP) 2003-11-26 EP disclosed
WO-2002068586-A2 HIV/FIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2002-09-06 WO disclosed
EP-1185869-A2 LIGAND-ANCHOR CONJUGATES FOR PRODUCING A BIOSENSOR LAYER Graffinity Pharmaceutical Design GmbH (DE) 2002-03-13 EP disclosed
CN-1330076-A Endothelin antagon INST OF TOXIC MEDICINES PLA S (CN) 2002-01-09 CN disclosed
CN-1330077-A Endothelin antegon INST OF TOXIC MEDICINES PLA S (CN) 2002-01-09 CN disclosed
WO-2000073796-A2 LIGAND-ANCHOR CONJUGATES FOR PRODUCING A BIOSENSOR LAYER GRAFFINITY PHARMACEUTICAL DESIGN GMBH (DE) 2000-12-07 WO disclosed
US-5364850-A Analgesics G. D. SEARLE & CO. (US) 1994-11-15 US disclosed
US-5272175-A Substituted tyrosyl diamide compounds G. D. SEARLE & CO. (US) 1993-12-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230257388-A1 GRANZYME B DIRECTED IMAGING AND THERAPY GZMB, PRF1, CTSB ALDH1A1 4592/4885LMNA 783/4885ACE 1545/4885
US-20200369673-A1 GRANZYME B DIRECTED IMAGING AND THERAPY GZMB, PRF1, CTSB ALDH1A1 4592/4885LMNA 783/4885ACE 1545/4885
US-11667645-B2 Granzyme B directed imaging and therapy GZMB, PRF1, CTSB ALDH1A1 4592/4885LMNA 783/4885ACE 1545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.