SCHEMBL6002435

SCHEMBL6002435

[CH2]C(CCCC)c1nc(C)sc1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.45
COMT P21964 4/20 0.38
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GCGR P47871 1/20 0.35
TSHR P16473 1/20 0.35
NR1H3 Q13133 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
HPGD P15428 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003294 0.78 ATP4A (0.43) COMTKDM4ENPC1ALDH1A1LMNA
SCHEMBL5547301 0.76 ALOX5 (0.46) ALOX5COMTPTGS1PTGS2KDM4E
SCHEMBL10242340 0.74 ALOX5 (0.58) ALOX5COMTPTGS1PTGS2KDM4E
SCHEMBL10242344 0.72 ALOX5 (0.51) ALOX5COMTPTGS1PTGS2KDM4E
SCHEMBL27629514 0.71 ALOX5 (0.50) ALOX5COMTPTGS1PTGS2KDM4E
SCHEMBL2093674 0.69 ALOX5 (0.56) ALOX5COMTPTGS1PTGS2NPC1
SCHEMBL2090158 0.68 ALOX5 (0.50) ALOX5COMTPTGS1PTGS2KDM4E
SCHEMBL6003969 0.68 ADORA3 (0.34) GCGRTSHRNR1H3
SCHEMBL10242337 0.67 ALOX5 (0.58) ALOX5COMTPTGS1PTGS2NPC1
SCHEMBL5167355 0.67 CYP17A1 (0.49) ALOX5PTGS2KDM4ESMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed