SCHEMBL6002979

SCHEMBL6002979

O=[C]N(c1ccccc1)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.32
NR1H3 Q13133 3/20 0.31
NR1H2 P55055 1/20 0.31
MEN1 O00255 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3486119 0.79 CES1 (0.37) NR1H3NR1H2MEN1CYP3A4CYP2C9
SCHEMBL6002568 0.69 TACR1 (0.30)
SCHEMBL6002270 0.68 NPSR1 (0.38) NR1H3NR1H2MEN1CYP3A4CYP2C9
SCHEMBL6792995 0.65 MEN1 (0.37) NR1H3NR1H2MEN1KMT2AALDH1A1
SCHEMBL2015505 0.63 ALDH1A1 (0.39) MEN1CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL28816160 0.63 ALDH1A1 (0.39) MEN1CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL12574813 0.63 ALDH1A1 (0.38) NR1H3NR1H2MEN1CYP3A4CYP2C9
SCHEMBL6790778 0.63 NR1H2 (0.32) NR1H3NR1H2ALDH1A1
SCHEMBL11871425 0.63 MLYCD (0.37) SMN1; SMN2NPSR1ALDH1A1ALOX15
SCHEMBL104821 0.62 ALDH1A1 (0.42) MEN1CYP3A4CYP2C9CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102532162-A 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMA CO LTD 2012-07-04 CN disclosed
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed