SCHEMBL6004285

SCHEMBL6004285

Cc1ccc(Oc2ccnc3ccc(OCc4ccccc4)cc23)c(-c2ncccn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
IP6K1 Q92551 1/20 0.42
DYRK1A Q13627 1/20 0.39
PLAU P00749 1/20 0.39
PLAT P00750 1/20 0.39
MAOA P21397 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NMT1 P30419 2/20 0.38
NMT2 O60551 1/20 0.38
ALOX5 P09917 1/20 0.38
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004827 0.90 CYP3A4 (0.44) CYP3A4IP6K1DYRK1APLAUPLAT
SCHEMBL6004179 0.88 CYP3A4 (0.44) CYP3A4IP6K1PLAUPLATNPC1
SCHEMBL6004895 0.87 CYP3A4 (0.45) CYP3A4IP6K1DYRK1APLAUPLAT
SCHEMBL6004162 0.84 ALDH1A1 (0.36) ALDH1A1HSD17B10SYKAURKBINCENP
SCHEMBL6005366 0.84 PDGFRB (0.36) SYKAURKBINCENP
SCHEMBL6004262 0.84 ALDH1A1 (0.36) CYP3A4KDM4EALDH1A1CYP1A2HSD17B10
SCHEMBL6004922 0.84 SLC22A12 (0.39) MAOAALDH1A1HSD17B10SYKAURKB
SCHEMBL6005251 0.84 PDE2A (0.39) ALDH1A1HSD17B10AURKB
SCHEMBL6005281 0.82 DDR2 (0.34)
SCHEMBL6004146 0.82 SRC (0.38) MEN1KMT2AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed