SCHEMBL6004317

SCHEMBL6004317

OC1=Nc2ccccc2CN1C1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.47
HTR2A P28223 5/20 0.47
CTSD P07339 3/20 0.47
PARP1 P09874 2/20 0.44
HTR2B P41595 5/20 0.43
BCHE P06276 3/20 0.42
ACHE P22303 2/20 0.42
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14498123 0.82 CTSD (0.70) HTR2CHTR2ACTSDPARP1HTR2B
SCHEMBL5386800 0.79 PARP1 (0.43) HTR2CHTR2APARP1HTR2B
SCHEMBL1976916 0.72 PARP1 (0.56) HTR2CHTR2APARP1HTR2B
SCHEMBL14417169 0.72 DRD2 (0.39) HTR2CHTR2ACTSDPARP1
SCHEMBL7985474 0.71 HTR2C (0.50) HTR2CHTR2APARP1HTR2BSIGMAR1
SCHEMBL28229327 0.71 NPC1 (0.44) HTR2CHTR2ACTSDPARP1HTR2B
SCHEMBL9280480 0.69 HTR2C (0.56) HTR2CHTR2APARP1HTR2B
SCHEMBL2210808 0.69 PARP1 (0.49) HTR2CHTR2APARP1HTR2BACHE
SCHEMBL30658421 0.69 PARP1 (0.49) HTR2CHTR2APARP1HTR2BACHE
SCHEMBL14608794 0.68 SIGMAR1 (0.43) CTSDBCHEACHEPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641781-A2 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2006-04-05 EP disclosed
WO-2005000807-A2 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2005-01-06 WO disclosed