SCHEMBL9280480

SCHEMBL9280480

c1ccc2c(c1)Cc1ccccc1N(C1CCNCC1)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 11/20 0.56
HTR2A P28223 7/20 0.56
HTR2B P41595 8/20 0.56
PARP1 P09874 3/20 0.43
CYP3A4 P08684 3/20 0.37
CYP2C9 P11712 2/20 0.37
HRH3 Q9Y5N1 1/20 0.37
LMNA P02545 2/20 0.36
CYP2D6 P10635 2/20 0.36
CHRM2 P08172 2/20 0.36
ADRA2A P08913 2/20 0.36
CHRM1 P11229 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
CHRM3 P20309 2/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
KCNH2 Q12809 2/20 0.36
MEN1 O00255 2/20 0.36
TP53 P04637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11103752 0.81 HTR2A (0.49) HTR2CHTR2AHTR2BCYP3A4CYP2C9
SCHEMBL2210808 0.81 PARP1 (0.49) HTR2CHTR2AHTR2BPARP1NAMPT
SCHEMBL30658421 0.81 PARP1 (0.49) HTR2CHTR2AHTR2BPARP1NAMPT
Hydrochloric Acid SCHEMBL3888469 0.79 PARP1 (0.48) HTR2CHTR2AHTR2BPARP1NAMPT
SCHEMBL11247722 0.78 HTR2C (0.50) HTR2CHTR2AHTR2BPARP1MEN1
SCHEMBL11242393 0.77 HTR2C (0.49) HTR2CHTR2AHTR2BPARP1
SCHEMBL11247293 0.77 HTR2C (0.49) HTR2CHTR2AHTR2BPARP1
SCHEMBL7985474 0.77 HTR2C (0.50) HTR2CHTR2AHTR2BPARP1HRH3
SCHEMBL2709111 0.77 HTR2C (0.77) HTR2CHTR2AHTR2BCYP2D6CHRM2
Hydrochloric Acid SCHEMBL3947175 0.75 HTR2C (0.75) HTR2CHTR2AHTR2BCYP2D6CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5461047-A Analgesics and treats prostaglandin-E2 mediated diseases in animals G. D. SEARLE & CO. (US) 1995-10-24 US disclosed
US-5354747-A Analgesics G. D. SEARLE & CO. (US) 1994-10-11 US disclosed
US-4434171-A NEUROLEPTIC, ANTIDEPRESSANT SANDOZ LTD. (CH) 1984-02-28 US disclosed