SCHEMBL6004768

SCHEMBL6004768

Oc1cc2cccnc2nc1-c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.51
L3MBTL1 Q9Y468 4/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MAPK14 Q16539 1/20 0.48
PDGFRB P09619 2/20 0.41
PDGFRA P16234 2/20 0.41
EGFR P00533 1/20 0.41
ALDH1A1 P00352 2/20 0.38
DAO P14920 1/20 0.38
HPGD P15428 1/20 0.38
MMP2 P08253 1/20 0.38
CHRM1 P11229 1/20 0.38
TSHR P16473 1/20 0.38
COMT P21964 1/20 0.38
ADRA1A P35348 1/20 0.38
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
QDPR P09417 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1692394 0.88 DHODH (0.44) KDM4EL3MBTL1NPC1RAB9AALDH1A1
SCHEMBL6004845 0.84 MAPK14 (0.52) KDM4ENPC1RAB9AMAPK14ALDH1A1
SCHEMBL6004749 0.84 CYP1A2 (0.41) KDM4EL3MBTL1NPC1RAB9AMAPK14
SCHEMBL6004302 0.84 KDM4E (0.43) KDM4EL3MBTL1NPC1RAB9AMAPK14
SCHEMBL3892242 0.84 COMT (0.43) KDM4EL3MBTL1ALDH1A1HPGDCOMT
SCHEMBL6004865 0.84 L3MBTL1 (0.54) KDM4EL3MBTL1NPC1RAB9APDGFRB
SCHEMBL6004176 0.80 SLC22A12 (0.41)
SCHEMBL3896975 0.77 KDM4E (0.45) KDM4EL3MBTL1NPC1RAB9AALDH1A1
SCHEMBL6002944 0.76 AURKA (0.53) KDM4EALDH1A1HPGDHDAC8
SCHEMBL30060806 0.76 KDM4E (0.43) KDM4EL3MBTL1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed