SCHEMBL6015050

SCHEMBL6015050

CN1C=C2C(=O)N(C3CCN(C(=O)[C@@H](Cc4ccc(OCc5ccccc5)cc4)NC(=O)O)CC3)CN2C1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 13/20 0.45
CACNA1B Q00975 3/20 0.42
ACE P12821 2/20 0.42
CALCRL Q16602 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451041 0.92 ALDH1A1 (0.43) CALCRL
SCHEMBL6015065 0.92 ALDH1A1 (0.43) CALCRL
SCHEMBL3450767 0.89 FPR2 (0.45) YAP1CACNA1B
SCHEMBL6015142 0.85 FPR2 (0.42) YAP1CALCRL
SCHEMBL6015116 0.83 CYP51A1 (0.42) ACECALCRL
SCHEMBL6015112 0.80 CCR1 (0.38)
SCHEMBL3449290 0.80 FPR2 (0.49)
SCHEMBL3449020 0.80 FPR2 (0.49)
SCHEMBL3448805 0.80 FPR2 (0.49)
SCHEMBL3449487 0.79 MAPT (0.37) YAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1695961-A1 UREA DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Pharmaceutical Company Limited (JP) 2006-08-30 EP disclosed