SCHEMBL6015116

SCHEMBL6015116

CN1C=C2C(=O)N(C3CCN(C(=O)[C@@H](Cc4cccnc4)NC(=O)O)CC3)CN2C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP51A1 Q16850 1/20 0.42
CHRM1 P11229 1/20 0.42
ACE P12821 2/20 0.39
F2 P00734 1/20 0.38
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
CALCA P06881 3/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CALCRL Q16602 2/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
RAMP1 O60894 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
FPR2 P25090 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015065 0.91 ALDH1A1 (0.43) CYP51A1CHRM1KDM4ESMN1; SMN2HSD17B10
SCHEMBL3451041 0.91 ALDH1A1 (0.43) CYP51A1CHRM1KDM4ESMN1; SMN2HSD17B10
SCHEMBL3449415 0.87 CYP51A1 (0.44) CYP51A1CHRM1ALDH1A1FPR2
SCHEMBL6015050 0.83 YAP1 (0.45) ACECALCRL
SCHEMBL6015142 0.83 FPR2 (0.42) CALCACALCRLFPR2
SCHEMBL6015112 0.82 CCR1 (0.38) KDM4EFPR2
SCHEMBL6015073 0.81 CCR1 (0.40)
SCHEMBL6015029 0.81 CCR1 (0.40) KDM4EHSD17B10CALCRLCTSBCTSS
SCHEMBL6015003 0.79 CCKBR (0.40) ACE
SCHEMBL3451164 0.78 ALDH1A1 (0.34) CHRM1PARP1PARP2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1695961-A1 UREA DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Pharmaceutical Company Limited (JP) 2006-08-30 EP disclosed