SCHEMBL6015618

SCHEMBL6015618

Cc1[c]cn(CC(=O)NCCN2CCCC2)n1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 4/20 0.43
CYP2D6 P10635 2/20 0.43
KDM4E B2RXH2 2/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TSHR P16473 2/20 0.42
MEN1 O00255 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015956 0.89 POLB (0.52) KMT2AKDM4EPOLBGAASMN1; SMN2
SCHEMBL6016081 0.84 TSHR (0.52) KMT2ANPSR1ALDH1A1CYP2D6KDM4E
SCHEMBL6015745 0.77 KDM4E (0.46) NPSR1ALDH1A1CYP2D6KDM4EPOLB
SCHEMBL15495602 0.74 KMT2A (0.45) KMT2ANPSR1ALDH1A1CYP2D6KDM4E
SCHEMBL4283848 0.70 ALDH1A1 (0.81) KMT2ANPSR1ALDH1A1KDM4EPOLB
SCHEMBL6016084 0.70 HDAC4 (0.34)
SCHEMBL15495676 0.69 CYP2D6 (0.47) KMT2AALDH1A1CYP2D6KDM4EPOLB
SCHEMBL7615075 0.69 TBXAS1 (0.40)
SCHEMBL2067370 0.69 POLB (0.46) KMT2AALDH1A1POLBMAPK1SMN1; SMN2
SCHEMBL6015620 0.68 HTT (0.50) KMT2ACYP2D6KDM4EPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed