SCHEMBL6015694

SCHEMBL6015694

O=C(c1ccc2[c]c[nH]c2c1)N1CCN(CCO)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
POLB P06746 2/20 0.49
HTT P42858 1/20 0.46
MAPK14 Q16539 2/20 0.44
AKR1C3 P42330 1/20 0.44
NAMPT P43490 1/20 0.43
TLR9 Q9NR96 1/20 0.43
TLR8 Q9NR97 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
PARP1 P09874 3/20 0.42
ALPL P05186 1/20 0.41
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
DUSP3 P51452 2/20 0.40
PTPN5 P54829 2/20 0.40
PTPN11 Q06124 2/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015723 0.87 PARP1 (0.48) ALDH1A1MAPK14PARP1DRD2
SCHEMBL6015819 0.86 ALDH1A1 (0.48) ALDH1A1POLBMAPK14TLR9TLR8
SCHEMBL6015833 0.85 KMT2A (0.52) ALDH1A1POLBCYP2D6CYP2C19MAPT
SCHEMBL6015913 0.81 SIGMAR1 (0.49) TLR9TLR8TLR7PARP1HPGD
SCHEMBL6015947 0.81 POLB (0.53) POLBTLR9TLR8TLR7HPGD
SCHEMBL6015825 0.80 SPIN1 (0.48)
SCHEMBL6015641 0.76 PDE3B (0.46) ALDH1A1HTTPDE3BPDE3AMAPT
SCHEMBL6015774 0.74 MAPK14 (0.42) ALDH1A1POLBHTTMAPK14AKR1C3
SCHEMBL6015942 0.74 L3MBTL3 (0.61) ALDH1A1
SCHEMBL6015966 0.72 HTR3A (0.54) ALDH1A1POLBPARP1CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed