SCHEMBL6016013

SCHEMBL6016013

CCN(CC)CCNCC(=O)c1ccc2[c]c[nH]c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
KDM4E B2RXH2 3/20 0.37
LMNA P02545 3/20 0.37
MAPK1 P28482 2/20 0.37
SLC22A2 O15244 1/20 0.37
SLC22A1 O15245 1/20 0.37
TSHR P16473 1/20 0.37
ACHE P22303 1/20 0.37
CYP2C19 P33261 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
BLM P54132 2/20 0.36
PMP22 Q01453 1/20 0.36
NFKB1 P19838 1/20 0.35
KCNH2 Q12809 1/20 0.35
POLB P06746 2/20 0.34
CYP3A4 P08684 1/20 0.34
THRB P10828 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015845 0.83 KDM4E (0.31) ALDH1A1KDM4EPOLBHPGDHTT
SCHEMBL6015884 0.80 HPGD (0.39) ALDH1A1KDM4ETSHRSMN1; SMN2GAA
SCHEMBL6015894 0.79 ALDH1A1 (0.42) ALDH1A1KDM4ELMNACYP2C19POLB
SCHEMBL6015672 0.79 EPHX1 (0.33) ALDH1A1KMT2AHPGD
SCHEMBL6015656 0.77 ALDH1A1 (0.39) ALDH1A1LMNAMAPK1TSHRPOLB
SCHEMBL6016047 0.77 HTR3A (0.39) ALDH1A1KDM4EPOLBGAAHSD17B10
SCHEMBL6015948 0.76 HTR3A (0.41) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL6016011 0.74 TSHR (0.32) ALDH1A1LMNAMAPK1SLC22A2SLC22A1
SCHEMBL6015748 0.74 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAMAPK1POLB
SCHEMBL6015811 0.71 ALDH1A1 (0.47) ALDH1A1KDM4ELMNASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed