SCHEMBL6016017

SCHEMBL6016017

OC1CCN(Cc2c[nH]c3[c]cccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.49
DRD4 P21917 4/20 0.49
DRD3 P35462 4/20 0.49
CYP2D6 P10635 2/20 0.47
BCHE P06276 1/20 0.47
LMNA P02545 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 1/20 0.43
MAPT P10636 1/20 0.43
JAK2 O60674 1/20 0.43
RAB9A P51151 1/20 0.43
HTR6 P50406 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
KRAS P01116 1/20 0.40
SOS1 Q07889 1/20 0.40
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015887 0.85 LMNA (0.59) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015775 0.84 LMNA (0.61) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015736 0.83 ALDH1A1 (0.54) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6016030 0.82 BCHE (0.49) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015640 0.82 BCHE (0.51) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015944 0.82 BCHE (0.48) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015685 0.82 HTR6 (0.63) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL6015714 0.77 HTR6 (0.58) DRD2DRD4DRD3CYP2D6BCHE
SCHEMBL27631244 0.69 HTR2C (0.44) CYP2D6KDM4EHTTHTR6ALDH1A1
SCHEMBL27883990 0.66 MPO (0.72) BCHEKDM4EMAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed