SCHEMBL6016049

SCHEMBL6016049

CN(C)CCCNC(=O)Cn1c[c]c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
P2RX4 Q99571 1/20 0.43
ALOX15 P16050 2/20 0.42
KDM4E B2RXH2 4/20 0.42
CYP1A2 P05177 1/20 0.41
TSHR P16473 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
DNM1 Q05193 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27620291 0.82 KDM4E (0.34) KDM4ECYP1A2TSHRSMN1; SMN2ALDH1A1
SCHEMBL4168685 0.81 GRIN1 (0.44) TSHRSMN1; SMN2
SCHEMBL6015764 0.76 PRKCA (0.42) KDM4ECYP1A2TSHRSMN1; SMN2MAPT
SCHEMBL17956205 0.72 HTR2C (0.51) CYP1A2ALDH1A1
SCHEMBL10397184 0.68 PTGS2 (0.57) HTTALOX15KDM4ESMN1; SMN2MAPT
SCHEMBL6015850 0.67 DNM1 (0.44) HTTP2RX4ALOX15KDM4ETSHR
SCHEMBL6015870 0.67 ALDH1A1 (0.54) HTTKDM4ECYP1A2TSHRSMN1; SMN2
SCHEMBL1557707 0.66 DNM1 (0.43) P2RX4ALOX15KDM4ETSHRMAPT
SCHEMBL7617275 0.66 KDM4E (0.46) P2RX4ALOX15KDM4EALDH1A1CYP2C9
SCHEMBL7093719 0.65 CNR1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed