SCHEMBL6016466

SCHEMBL6016466

O=C(O)c1cnc(Cn2ccnc2)nc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 12/20 0.51
CYP11B2 P19099 11/20 0.51
CYP19A1 P11511 4/20 0.48
NTRK1 P04629 1/20 0.47
TBXAS1 P24557 1/20 0.47
CYP17A1 P05093 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016363 0.76 LMNA (0.46) NTRK1
SCHEMBL6016407 0.75 KDM4E (0.48)
SCHEMBL6016399 0.75 ALDH1A1 (0.49)
SCHEMBL6016362 0.73 PTGS2 (0.45)
SCHEMBL6016324 0.73 CHRM5 (0.46) NTRK1
SCHEMBL27488851 0.72 LMNA (0.43)
SCHEMBL6016349 0.72 NTRK1 (0.45) NTRK1
SCHEMBL28416685 0.72 CYP19A1 (0.76) CYP11B1CYP11B2CYP19A1TBXAS1
SCHEMBL6016470 0.71 NTRK1 (0.42) NTRK1
SCHEMBL6016450 0.71 MEN1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
CN-1166643-C 4-phenyl-pyrimidine derivatives - 2004-09-15 CN disclosed
CN-1353697-A 4-phenyl-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2002-06-12 CN disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed