SCHEMBL6017086

SCHEMBL6017086

CC(C)(C)OC(=O)c1cc[nH]c1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
PREP P48147 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GABRA1 P14867 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
GABRA2 P47869 2/20 0.31
GABRA4 P48169 2/20 0.31
GABRA6 Q16445 2/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1320587 0.76 ELANE (0.32) ADRA1AADRA1BGABRA1GABRG2GABRB3
SCHEMBL18703898 0.74 ADRA1A (0.34) ADRA1AADRA1BCYP2C9CYP2C19NPSR1
SCHEMBL15567828 0.73 RAB9A (0.38) ADRA1AADRA1BCYP2C9CYP2C19NPSR1
SCHEMBL1566864 0.73 CA12 (0.38) ADRA1AADRA1BGABRA1GABRG2GABRB3
SCHEMBL163017 0.73 CA12 (0.35) ADRA1AADRA1BGABRA1GABRG2GABRB3
SCHEMBL8562952 0.71 ALDH1A1 (0.38) ADRA1AADRA1BGABRA1GABRG2GABRB3
SCHEMBL624330 0.69 RAB9A (0.33) ADRA1AADRA1BGABRA1GABRG2GABRB3
SCHEMBL28587355 0.69 ALDH1A1 (0.36) ADRA1AADRA1BNPSR1ALDH1A1AR
SCHEMBL28816343 0.69 ALDH1A1 (0.45) ADRA1AADRA1BLMNAALDH1A1RAB9A
SCHEMBL3801958 0.67 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2MAPTALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660443-A2 CYCLIC AMINE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT SCHERING CORPORATION (US) 2006-05-31 EP disclosed
WO-2005016876-A2 CYCLIC AMINE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT SCHERING CORPORATION (US) 2005-02-24 WO disclosed