SCHEMBL6017182

SCHEMBL6017182

CCOC(=O)Cc1c[nH]c2cccc(OCCc3ccc(-c4ccc(C(F)(F)F)cc4)nc3C)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
POLB P06746 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARG P37231 3/20 0.37
PPARA Q07869 3/20 0.37
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADRB2 P07550 1/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5617095 0.92 KDM4E (0.40) KMT2AMEN1POLBPPARGPPARA
SCHEMBL4432117 0.77 PPARG (0.50) KMT2AMEN1SMN1; SMN2HPGDHTT
SCHEMBL6052553 0.76 PPARD (0.54) PPARGPPARAPPARD
SCHEMBL6017246 0.76 PPARG (0.43) PPARGPPARAPPARD
SCHEMBL6017372 0.75 PKM (0.43) PKMPPARGPPARATRPV1PPARD
SCHEMBL6017241 0.75 PPARG (0.35) PPARGPPARAL3MBTL1TRPV1PPARD
SCHEMBL4421601 0.74 TRPM2 (0.43) PPARGPPARAALDH1A1L3MBTL1SYK
SCHEMBL6052560 0.74 PPARD (0.54) PPARGPPARAMAPTPPARD
SCHEMBL5673680 0.74 PPARD (0.51) PPARGPPARAALDH1A1L3MBTL1PPARD
SCHEMBL6017148 0.74 TRPV1 (0.44) PPARGPPARAMTNR1AMTNR1BTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed