SCHEMBL6017230

SCHEMBL6017230

CCOC(=O)Cc1c[nH]c2cc(OCCc3cnc(-c4ccc(C(F)(F)F)cc4)nc3C3CC3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
PPARA Q07869 4/20 0.37
PPARG P37231 3/20 0.37
MAOB P27338 2/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
FOS P01100 1/20 0.35
JUN P05412 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
PPARD Q03181 1/20 0.34
KCNH2 Q12809 1/20 0.33
TRPC3 Q13507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017580 0.93 MAOB (0.40) PKMPPARAMAOBTDP1FOS
SCHEMBL6017141 0.90 PPARA (0.39) PPARAPPARGTRPV1PPARD
SCHEMBL6017387 0.87 TRPV1 (0.40) PKMPPARAPPARGMAOBTRPV1
SCHEMBL5617383 0.83 PPARD (0.43) PPARAPPARGMAOBPPARD
SCHEMBL5668158 0.81 PPARD (0.48) PPARAPPARGPPARD
SCHEMBL6028937 0.79 GRIN2B (0.41) PPARAPPARGMAOBMAPTFOS
SCHEMBL6017371 0.78 TRPV1 (0.45) PKMPPARAPPARGMAOBLMNA
SCHEMBL6065376 0.77 PKM (0.41) PKMPPARAPPARGLMNAMEN1
SCHEMBL6017575 0.77 TRPV1 (0.46) PKMPPARAPPARGMAOBLMNA
SCHEMBL6017240 0.77 KDM4E (0.43) PPARAPPARGLMNAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed