SCHEMBL6020904

SCHEMBL6020904

N#CN(CC(N)=O)C(=O)[CH]Cc1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.41
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
HSP90AA1 P07900 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPK1 P28482 1/20 0.32
CAMK2A Q9UQM7 1/20 0.32
EGFR P00533 1/20 0.32
ERBB2 P04626 1/20 0.32
SLC7A5 Q01650 1/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
ABAT P80404 1/20 0.31
ESR1 P03372 4/20 0.30
ESR2 Q92731 4/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
THRB P10828 1/20 0.30
CISD1 Q9NZ45 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6020762 0.87 MCL1 (0.36) CA2CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL6020719 0.80 CYP1A2 (0.36) CA2CYP1A2
SCHEMBL6019621 0.79 CA2 (0.40) CA2CYP1A2CYP2C9CYP2C19CAMK2A
SCHEMBL4955729 0.71 CA2 (0.43) CA2CYP2C19CAMK2ASLC7A5ABAT
SCHEMBL2122257 0.70 CA2 (0.54) CA2CYP2C19CAMK2ASLC7A5MEN1
SCHEMBL6019641 0.70 CYP2A6 (0.42) CA2ALDH1A1
SCHEMBL6021610 0.70 MAPT (0.42) MEN1KMT2AALDH1A1CYP3A4
SCHEMBL6021436 0.66 ALDH1A1 (0.37) CA2CYP1A2CYP2C19EGFRALDH1A1
SCHEMBL8067640 0.65 CA2 (0.52) CA2CAMK2ASLC7A5MEN1KMT2A
SCHEMBL5215999 0.64 CA2 (0.55) CA2CYP2C19CAMK2ASLC7A5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060252813-A1 Apparatus for curing a composite laminate JERINI AG (DE) 2006-11-09 US claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1433778-A1 Use of nitriles as rotamase inhibitors Jerini AG (DE) 2004-06-30 EP claimed
EP-1433779-A1 Use of nitriles as inhibitors of non-proteolytic enzymes Jerini AG (DE) 2004-06-30 EP claimed
US-20060252813-A1 Apparatus for curing a composite laminate JERINI AG (DE) 2006-11-09 US disclosed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed
EP-1433778-A1 Use of nitriles as rotamase inhibitors Jerini AG (DE) 2004-06-30 EP disclosed
EP-1433779-A1 Use of nitriles as inhibitors of non-proteolytic enzymes Jerini AG (DE) 2004-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060252813-A1 Apparatus for curing a composite laminate DHX29, HDHD5, DHRS9 CA2 2390/4885CYP1A2 3116/4885CYP2C9 2146/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.