SCHEMBL6028353

SCHEMBL6028353

CCOC(C(=O)NCc1ccc(C#N)cc1O)N1C=C2C=CC(=O)C(C)=C2C1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.33
ENPP2 Q13822 1/20 0.31
SETDB1 Q15047 1/20 0.31
DRD2 P14416 3/20 0.31
DRD3 P35462 3/20 0.31
DRD4 P21917 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028546 0.87 F10 (0.33) ENPP2
SCHEMBL6028074 0.86 SLC1A2 (0.34) ENPP2
SCHEMBL6028367 0.75 ST14 (0.39)
Acetic Acid SCHEMBL6027976 0.73 F10 (0.43)
SCHEMBL6028623 0.73 P2RX7 (0.34) P2RX7
SCHEMBL6078343 0.73 SDCBP (0.34) P2RX7SETDB1DRD2DRD3DRD4
SCHEMBL6078352 0.73 SDCBP (0.34) P2RX7SETDB1DRD2DRD3DRD4
SCHEMBL6079105 0.70 LMNA (0.40) DRD2DRD3DRD4
SCHEMBL6079096 0.70 LMNA (0.40) DRD2DRD3DRD4
SCHEMBL6029054 0.69 F10 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706396-A1 N-(4-CARBAMIMIDOYL-BENZYL)-2-ALKOXY-2-HETEROCYCLYL ACETAMIDES AS INHIBITORS OF THE FORMATION OF COAGULATION FACTORS XA, IXA AND THROMBIN INDUCED BY FACTOR VIIA F.HOFFMANN-LA ROCHE AG (CH) 2006-10-04 EP disclosed
WO-2005058868-A1 N-(4-CARBAMIMIDOYL-BENZYL) -2-ALKOXY-2-HETEROCYCLYL ACETAMIDES AS INHIBITORS OF THE FORMATION OF COAGULATION FACTORS XA, IXA AND THROMBIN INDUCED BY FACTOR VIIA F. HOFFMANN-LA ROCHE AG (CH) 2005-06-30 WO disclosed