SCHEMBL6028513

SCHEMBL6028513

COc1cccc(-c2cnc(OCC(=O)NC(Cc3cccc(Cl)c3Cl)C3CCCNC3)nc2)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.41
GRIN2B Q13224 3/20 0.41
CHEK1 O14757 2/20 0.39
DGAT2 Q96PD7 1/20 0.39
CDK9 P50750 3/20 0.37
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CTSA P10619 1/20 0.35
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030272 0.92 CHEK1 (0.37) GRIN1GRIN2BCHEK1CDK9CYP3A4
SCHEMBL6029742 0.90 CDK9 (0.38) CDK9SLC6A2SLC6A4
SCHEMBL6029349 0.89 MAPK1 (0.38) CDK9CYP3A4SLC6A2SLC6A4TP53
SCHEMBL6030392 0.88 CHEK1 (0.41) GRIN1GRIN2BCHEK1CDK9CYP2C19
SCHEMBL7826595 0.88 SLC6A4 (0.39) GRIN1GRIN2BCYP3A4SLC6A2SLC6A4
SCHEMBL6030283 0.81 GHSR (0.37) GRIN1GRIN2BCHEK1CDK9CYP3A4
SCHEMBL7831249 0.81 SLC6A4 (0.38) CYP3A4SLC6A2SLC6A4
SCHEMBL6028530 0.81 CHEK1 (0.37) GRIN1GRIN2BCHEK1CDK9CYP3A4
SCHEMBL6030139 0.79 ALOX15 (0.37) CDK9SLC6A2SLC6A4MAPT
SCHEMBL6029151 0.79 CHEK1 (0.39) GRIN1GRIN2BCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed