SCHEMBL7826595

SCHEMBL7826595

COc1ccc(-c2cnc(OCC(=O)NC(Cc3cccc(Cl)c3Cl)C3CCNC3)nc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.39
SLC6A2 P23975 5/20 0.39
MBTPS1 Q14703 2/20 0.38
SLC6A3 Q01959 4/20 0.38
CYP2D6 P10635 2/20 0.38
KCNH2 Q12809 2/20 0.38
CYP3A4 P08684 1/20 0.38
CTSD P07339 1/20 0.37
AKT1 P31749 1/20 0.36
GRIN1 Q05586 4/20 0.36
GRIN2B Q13224 4/20 0.36
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030272 0.95 CHEK1 (0.37) SLC6A4SLC6A2MBTPS1SLC6A3CYP2D6
SCHEMBL7831249 0.90 SLC6A4 (0.38) SLC6A4SLC6A2MBTPS1SLC6A3CYP2D6
SCHEMBL7818522 0.88 SLC6A4 (0.38) SLC6A4SLC6A2MBTPS1SLC6A3CYP2D6
SCHEMBL6028513 0.88 GRIN1 (0.41) SLC6A4SLC6A2CYP3A4GRIN1GRIN2B
SCHEMBL7829393 0.88 SLC6A4 (0.38) SLC6A4SLC6A2MBTPS1SLC6A3CYP2D6
SCHEMBL6029742 0.86 CDK9 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL7829880 0.85 AKT1 (0.42) SLC6A4SLC6A2SLC6A3CTSDAKT1
Hydrochloric Acid SCHEMBL7833338 0.84 AKT1 (0.42) SLC6A4SLC6A2SLC6A3CTSDAKT1
SCHEMBL6029349 0.84 MAPK1 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL6030283 0.84 GHSR (0.37) SLC6A4SLC6A2MBTPS1SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed