SCHEMBL6029102

SCHEMBL6029102

O=C(CSc1ncc(-c2ccccc2)cn1)NC(Cc1ccc(F)c(Cl)c1)C1CCCNC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.39
NTRK1 P04629 5/20 0.38
MAPK1 P28482 4/20 0.38
MC4R P32245 2/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
KAT7 O95251 1/20 0.35
KAT6A Q92794 1/20 0.35
KAT5 Q92993 1/20 0.35
CTSC P53634 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
SOS1 Q07889 1/20 0.35
CCNT1 O60563 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028919 0.94 CHEK1 (0.39) CHEK1NTRK1MC4RKAT7KAT6A
SCHEMBL6030280 0.93 NTRK1 (0.39) CHEK1NTRK1MC4RCTSCKMT2A
SCHEMBL6028983 0.93 CDK2 (0.38) CHEK1MAPK1MC4RGRIN2BALDH1A1
SCHEMBL6029095 0.90 CHEK1 (0.39) CHEK1MAPK1GRIN1GRIN2BALDH1A1
SCHEMBL6028900 0.89 CDK8 (0.36) CHEK1NTRK1MAPK1MC4RLMNA
SCHEMBL6029438 0.88 CHEK1 (0.39) CHEK1MAPK1GRIN1GRIN2BLMNA
SCHEMBL6030341 0.87 CHEK1 (0.36) CHEK1MC4RGAA
SCHEMBL6029129 0.86 CHEK1 (0.35) CHEK1MC4RALDH1A1LMNAGAA
SCHEMBL6028338 0.85 CHEK1 (0.40) CHEK1
SCHEMBL6028748 0.84 CHEK1 (0.39) CHEK1GRIN1GRIN2BALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed