SCHEMBL6028338

SCHEMBL6028338

O=C(CSc1ncc(-c2ccccc2)cn1)NC(Cc1ccc2cc[nH]c2c1)C1CCCNC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 7/20 0.40
MAPKAPK2 P49137 1/20 0.36
F2 P00734 1/20 0.35
PRKCZ Q05513 3/20 0.35
PRKD2 Q9BZL6 3/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
KCNH2 Q12809 1/20 0.35
CHEK2 O96017 2/20 0.34
MET P08581 2/20 0.34
F10 P00742 1/20 0.34
CCNK O75909 1/20 0.34
CDK7 P50613 1/20 0.34
CCNH P51946 1/20 0.34
MNAT1 P51948 1/20 0.34
CDK12 Q9NYV4 1/20 0.34
PDPK1 O15530 1/20 0.34
RPS6KB1 P23443 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030341 0.88 CHEK1 (0.36) CHEK1PRKCZPRKD2JAK1JAK3
SCHEMBL6028349 0.87 LMNA (0.41) CHEK1PDPK1
SCHEMBL6030280 0.87 NTRK1 (0.39) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6028983 0.87 CDK2 (0.38) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6029129 0.86 CHEK1 (0.35) CHEK1PRKCZPRKD2JAK1JAK3
SCHEMBL6028919 0.85 CHEK1 (0.39) CHEK1JAK1JAK3KCNH2
SCHEMBL6029102 0.85 CHEK1 (0.39) CHEK1
SCHEMBL6028900 0.83 CDK8 (0.36) CHEK1JAK1JAK3CCNKCDK7
SCHEMBL6028834 0.80 LMNA (0.42) CHEK1MAPKAPK2
SCHEMBL6029595 0.79 NPC1 (0.37) CHEK1JAK1JAK3KCNH2CCNK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed