SCHEMBL6030341

SCHEMBL6030341

O=C(CSc1ncc(-c2ccccc2)cn1)NC(Cc1ccc(O)c(O)c1)C1CCCNC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
KCNH2 Q12809 1/20 0.36
PBK Q96KB5 1/20 0.36
F10 P00742 1/20 0.35
PDPK1 O15530 1/20 0.35
RPS6KB1 P23443 1/20 0.35
PRKCZ Q05513 4/20 0.35
PRKD2 Q9BZL6 4/20 0.35
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
MRE11 P49959 1/20 0.34
MC4R P32245 1/20 0.34
MME P08473 1/20 0.33
ACE P12821 1/20 0.33
CPA1 P15085 1/20 0.33
ACE2 Q9BYF1 1/20 0.33
CDK2AP1 O14519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030280 0.89 NTRK1 (0.39) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6028983 0.89 CDK2 (0.38) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6029129 0.89 CHEK1 (0.35) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6028338 0.88 CHEK1 (0.40) CHEK1JAK1JAK3KCNH2F10
SCHEMBL6028919 0.87 CHEK1 (0.39) CHEK1JAK1JAK3KCNH2MC4R
SCHEMBL6029102 0.87 CHEK1 (0.39) CHEK1GAAMC4R
SCHEMBL6028900 0.85 CDK8 (0.36) CHEK1JAK1JAK3GAAMC4R
SCHEMBL6029595 0.81 NPC1 (0.37) CHEK1JAK1JAK3KCNH2GAA
SCHEMBL6029268 0.81 MAPT (0.43)
SCHEMBL6028842 0.80 CHEK1 (0.39) CHEK1PDPK1RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed