SCHEMBL6029129

SCHEMBL6029129

O=C(CSc1ncc(-c2ccccc2)cn1)NC(Cc1ccc2c(c1)CCC2)C1CCCNC1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.35
KCNH2 Q12809 2/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 3/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
F10 P00742 1/20 0.34
PDPK1 O15530 1/20 0.34
RPS6KB1 P23443 1/20 0.34
PRKCZ Q05513 3/20 0.34
PRKD2 Q9BZL6 3/20 0.34
MC4R P32245 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
HTR2C P28335 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030341 0.89 CHEK1 (0.36) CHEK1KCNH2JAK1JAK3F10
SCHEMBL6028983 0.88 CDK2 (0.38) CHEK1KCNH2JAK1JAK3LMNA
SCHEMBL6030280 0.88 NTRK1 (0.39) CHEK1KCNH2JAK1JAK3MAPT
SCHEMBL6028822 0.87 LMNA (0.40) CHEK1RAB9ALMNAMAPTHTT
SCHEMBL6028338 0.86 CHEK1 (0.40) CHEK1KCNH2JAK1JAK3F10
SCHEMBL6029102 0.86 CHEK1 (0.39) CHEK1LMNAALDH1A1MC4RGAA
SCHEMBL6028919 0.86 CHEK1 (0.39) CHEK1KCNH2JAK1JAK3MC4R
SCHEMBL6028900 0.84 CDK8 (0.36) CHEK1JAK1JAK3LMNAMAPT
SCHEMBL6029595 0.80 NPC1 (0.37) CHEK1KCNH2JAK1JAK3RAB9A
SCHEMBL6029268 0.79 MAPT (0.43) RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed