SCHEMBL6029595

SCHEMBL6029595

O=C(CSc1ncc(-c2ccccc2)cn1)NC(Cc1cccc(Cl)c1Cl)C1CCCNC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SLC6A2 P23975 5/20 0.36
SLC6A4 P31645 5/20 0.36
SLC6A3 Q01959 4/20 0.35
KCNH2 Q12809 3/20 0.35
CYP2D6 P10635 2/20 0.35
CYP3A4 P08684 1/20 0.35
NTRK1 P04629 1/20 0.35
CHEK1 O14757 2/20 0.34
JAK1 P23458 1/20 0.34
JAK3 P52333 1/20 0.34
CCNT1 O60563 2/20 0.34
CCNK O75909 2/20 0.34
CDK9 P50750 2/20 0.34
CDK12 Q9NYV4 2/20 0.34
CDK7 P50613 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028530 0.91 CHEK1 (0.37) NPC1HPGDRAB9ASLC6A2SLC6A4
SCHEMBL7829393 0.86 SLC6A4 (0.38) NPC1RAB9ASLC6A2SLC6A4SLC6A3
SCHEMBL6028983 0.85 CDK2 (0.38) HPGDMAPK1KCNH2CHEK1JAK1
SCHEMBL6028919 0.83 CHEK1 (0.39) KCNH2NTRK1CHEK1JAK1JAK3
SCHEMBL6029102 0.83 CHEK1 (0.39) HPGDMAPK1NTRK1CHEK1CCNT1
SCHEMBL6028900 0.81 CDK8 (0.36) MAPK1SMN1; SMN2NTRK1CHEK1JAK1
SCHEMBL6030341 0.81 CHEK1 (0.36) KCNH2CHEK1JAK1JAK3SIGMAR1
SCHEMBL6030280 0.80 NTRK1 (0.39) KCNH2NTRK1CHEK1JAK1JAK3
SCHEMBL6029129 0.80 CHEK1 (0.35) RAB9AKCNH2CHEK1JAK1JAK3
SCHEMBL6028338 0.79 CHEK1 (0.40) SLC6A2SLC6A4SLC6A3KCNH2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed