SCHEMBL6036284

SCHEMBL6036284

CNC(=O)N(N)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
AOC3 Q16853 1/20 0.48
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HDAC3 O15379 2/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC2 Q92769 2/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
LMNA P02545 1/20 0.44
ABCC1 P33527 1/20 0.43
TSHR P16473 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27831817 0.83 ALDH1A1 (0.49) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL6422289 0.82 NPC1 (0.47) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL19027679 0.81 ALDH1A1 (0.65) NPC1RAB9AALDH1A1NPSR1KMT2A
SCHEMBL22649239 0.80 ALDH1A1 (0.46) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL258776 0.80 AOC3 (0.54) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL13903505 0.80 PTGES (0.54) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL13903560 0.80 EPHX2 (0.48) HDAC3KMT2AMEN1
SCHEMBL968919 0.79 NPC1 (0.67) NPC1RAB9AKMT2AMEN1CA12
SCHEMBL22649147 0.79 HDAC3 (0.45) NPC1RAB9AAOC3ALDH1A1NPSR1
SCHEMBL10416109 0.79 AOC3 (0.54) NPC1RAB9AAOC3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644025-A4 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS VION PHARMACEUTICALS INC (US) 2006-11-15 EP disclosed
EP-1644025-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS Vion Pharmaceuticals, Inc. (US) 2006-04-12 EP disclosed
US-20050043244-A1 Water-soluble SHPs as novel alkylating agents VION PHARMACEUTICALS, INC. (US) 2005-02-24 US disclosed
US-6855695-B2 Water-soluble SHPs as novel alkylating agents VION PHARMACEUTICALS, INC. (US) 2005-02-15 US disclosed
WO-2005004897-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS VION PHARMACEUTICALS, INC. (US) 2005-01-20 WO disclosed
US-20040254103-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS NANOSHIFT, LLC 2004-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040254103-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS SHPRH, OGFR, COG3 NPC1 3841/4885RAB9A 3812/4885AOC3 2260/4885
US-20050043244-A1 Water-soluble SHPs as novel alkylating agents GRM3, GRIA3, SHPRH NPC1 4197/4885RAB9A 4320/4885AOC3 502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.