SCHEMBL6047597

SCHEMBL6047597

Cc1cccc(C2=CC(C(F)(F)F)=CC[CH]2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.38
PTPN5 P54829 1/20 0.36
ENPP1 P22413 1/20 0.35
SDHB P21912 1/20 0.35
PDK2 Q15119 1/20 0.33
NISCH Q9Y2I1 2/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
ACHE P22303 2/20 0.32
PTGS1 P23219 3/20 0.32
PTGS2 P35354 3/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
RAB9A P51151 2/20 0.32
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047587 0.83 HTR2C (0.42) TSHR
SCHEMBL6047625 0.82 HTR2C (0.35) PDK2CHRNB4CHRNA3ALDH1A1KMT2A
SCHEMBL4808466 0.76 ACHE (0.38) NISCHCHRNB4CHRNA3ACHEALDH1A1
SCHEMBL4804654 0.75 ACHE (0.39) NISCHCHRNB4CHRNA3ACHEALDH1A1
SCHEMBL6408167 0.72 MAPT (0.33) NISCHCHRNB4CHRNA3ACHEALDH1A1
SCHEMBL6900961 0.70 RAB9A (0.41) NISCHCHRNB4CHRNA3ACHEALDH1A1
SCHEMBL4014782 0.70 PGR (0.36) CHRNB4CHRNA3ALDH1A1
SCHEMBL5698918 0.67
SCHEMBL5887149 0.66 AR (0.38) ARPTPN5ENPP1SDHBPDK2
SCHEMBL5143915 0.66 ACHE (0.38) NISCHCHRNB4CHRNA3ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed