SCHEMBL6047604

SCHEMBL6047604

COc1ccc(-c2ccccc2C2=CC(Oc3ccccc3)=CC[CH]2)c2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.35
TTR P02766 3/20 0.35
EP300 Q09472 1/20 0.34
KAT8 Q9H7Z6 1/20 0.34
ALOX5 P09917 1/20 0.34
BRD4 O60885 2/20 0.33
NQO1 P15559 1/20 0.33
IMPDH2 P12268 1/20 0.33
IMPDH1 P20839 1/20 0.33
PRMT1 Q99873 1/20 0.32
MAPT P10636 2/20 0.32
LTA4H P09960 1/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 2/20 0.32
CDC25B P30305 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
PABPC1 P11940 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047599 0.88 IDO1 (0.39) IDO1EP300KAT8NQO1IMPDH2
SCHEMBL6047663 0.81 MAPT (0.35) TTRALOX5BRD4NQO1MAPT
SCHEMBL6047596 0.78 ABL1 (0.45) MAPTLTA4HKMT2AALDH1A1HTT
SCHEMBL6047648 0.74 NAAA (0.42) BRD4LTA4HADORA2A
SCHEMBL6047633 0.72 PTPN1 (0.36) MAPTLTA4HALDH1A1KDM4EMAPK1
SCHEMBL6047613 0.70 THRA (0.39) MAPTKDM4ELMNAADORA2AMAPK1
SCHEMBL6047602 0.70 NAAA (0.37) MAPTLTA4HKDM4EADORA2AMAPK1
SCHEMBL12019868 0.69 IDO1 (0.59) IDO1EP300KAT8NQO1IMPDH2
SCHEMBL12019937 0.69 IDO1 (0.59) IDO1EP300KAT8NQO1IMPDH2
SCHEMBL12019841 0.69 IDO1 (0.64) IDO1EP300KAT8NQO1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed