SCHEMBL6066477

SCHEMBL6066477

CN(C)CNS(=O)(=O)c1ccccc1-c1ccc(C=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAT1 P18440 1/20 0.42
OPRM1 P35372 2/20 0.41
OPRK1 P41145 2/20 0.41
DRD1 P21728 3/20 0.40
CASP1 P29466 2/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
FEN1 P39748 5/20 0.39
ALOX5AP P20292 4/20 0.39
GRIA4 P48058 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6066483 0.81 OPRM1 (0.43) OPRM1OPRK1FEN1ALOX5AP
SCHEMBL7617752 0.81 OPRM1 (0.43) OPRM1OPRK1FEN1ALOX5AP
SCHEMBL489577 0.77 ALOX5AP (0.55) NAT1FEN1ALOX5AP
SCHEMBL3221376 0.74 OPRM1 (0.54) NAT1OPRM1OPRK1DRD1CASP1
SCHEMBL7614739 0.73 AGTR2 (0.41)
SCHEMBL839417 0.71 DRD1 (0.46) NAT1DRD1CASP1DRD2DRD4
SCHEMBL7803455 0.71 DRD1 (0.46) NAT1DRD1DRD2DRD4DRD5
SCHEMBL6066470 0.71 LMNA (0.41) NAT1OPRM1OPRK1DRD1CASP1
SCHEMBL6066480 0.71 LMNA (0.41) NAT1OPRM1OPRK1DRD1CASP1
SCHEMBL8511462 0.71 LMNA (0.41) NAT1OPRM1OPRK1DRD1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067665-B2 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-06-27 US disclosed
US-6953857-B2 Oxybenzamide derivatives useful for inhibiting factor Xa or viia AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2005-10-11 US disclosed
US-20050165058-A1 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2005-07-28 US disclosed
EP-1349847-B1 OXYBENZAMIDES DERIVATIVES AS FACTOR XA INHIBITORS AVENTIS PHARMA GMBH (DE) 2005-04-20 EP disclosed
EP-1349847-A1 OXYBENZAMIDES DERIVATIVES AS FACTOR XA INHIBITORS Aventis Pharma Deutschland GmbH (DE) 2003-10-08 EP disclosed
US-20020198195-A1 New oxybenzamide derivatives useful for inhibiting factor Xa or VIIa SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2002-12-26 US disclosed
WO-2002051831-A1 OXYBENZAMIDES DERIVATIVES AS FACTOR XA INHIBITORS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-07-04 WO disclosed
EP-1217000-A1 Inhibitors of factor Xa and factor VIIa Aventis Pharma Deutschland GmbH (DE) 2002-06-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165058-A1 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla F12, F11, F5 NAT1 1652/4885OPRM1 189/4885OPRK1 378/4885
US-20020198195-A1 New oxybenzamide derivatives useful for inhibiting factor Xa or VIIa F9, F11, F5 NAT1 1185/4885OPRM1 302/4885OPRK1 369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.