SCHEMBL6074882

SCHEMBL6074882

FC(F)(F)c1ccc(C(S)(Cl)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.48
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ORAI1 Q96D31 1/20 0.42
ORAI2 Q96SN7 1/20 0.42
ORAI3 Q9BRQ5 1/20 0.42
TRPV6 Q9H1D0 1/20 0.42
MGLL Q99685 1/20 0.42
GSK3B P49841 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
AHR P35869 1/20 0.39
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL63468 0.78 ALDH1A1 (0.67) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL4471260 0.77 ALDH1A1 (0.50) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL10672363 0.77 ALDH1A1 (0.50) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL1508480 0.77 ALDH1A1 (0.50) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL11598948 0.77 ALDH1A1 (0.50) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL1539075 0.77 TSHR (0.50) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL7641117 0.72 ALDH1A1 (0.46) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL21566844 0.72 ALDH1A1 (0.46) KIF11ALDH1A1TSHRCES2CES1
SCHEMBL677928 0.72 ALDH1A1 (0.46) KIF11ALDH1A1TSHRCES2CES1
Iodide SCHEMBL29093539 0.72 ALDH1A1 (0.59) KIF11ALDH1A1TSHRCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067538-B2 MCP-1 receptor antagonists and methods of use thereof WARNER-LAMBERT COMPANY, LLC (US) 2006-06-27 US disclosed
US-20050171163-A1 MCP-1 receptor antagonists and methods of use thereof BRATTON LARRY D (US) 2005-08-04 US disclosed
EP-1539685-A1 MCP-1 RECEPTOR ANTAGONISTS AND METHOD OF USE THEREOF Warner-Lambert Company LLC (US) 2005-06-15 EP disclosed
WO-2004014847-A1 MCP-1 RECEPTOR ANTAGONISTS AND METHOD OF USE THEREOF WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171163-A1 MCP-1 receptor antagonists and methods of use thereof CCR2, CCR1, CCL2 KIF11 3752/4885ALDH1A1 565/4885TSHR 744/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.