SCHEMBL4471260

SCHEMBL4471260

FC(F)(F)c1ccc(C(Cl)(Cl)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50
KIF11 P52732 6/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
ORAI1 Q96D31 1/20 0.46
ORAI2 Q96SN7 1/20 0.46
ORAI3 Q9BRQ5 1/20 0.46
TRPV6 Q9H1D0 1/20 0.46
MGLL Q99685 1/20 0.46
GSK3B P49841 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
AHR P35869 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL63468 0.83 ALDH1A1 (0.67) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL10672363 0.81 ALDH1A1 (0.50) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL1539075 0.81 TSHR (0.50) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL1508480 0.81 ALDH1A1 (0.50) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL11598948 0.81 ALDH1A1 (0.50) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL6074882 0.77 KIF11 (0.48) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL7641117 0.77 ALDH1A1 (0.46) ALDH1A1TSHRKIF11CES2CES1
SCHEMBL677928 0.77 ALDH1A1 (0.46) ALDH1A1TSHRKIF11CES2CES1
Bromide SCHEMBL29093544 0.76 ALDH1A1 (0.59) ALDH1A1TSHRKIF11CES2CES1
Iodide SCHEMBL29093539 0.76 ALDH1A1 (0.59) ALDH1A1TSHRKIF11CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576088-B2 Benzodioxole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
EP-1532132-B1 NOVEL BENZODIOXOLES HOFFMANN LA ROCHE (CH) 2008-03-19 EP disclosed
US-20050143373-A1 Benzodioxole derivatives ALANINE ALEXANDER (FR) 2005-06-30 US disclosed
US-6900227-B2 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. (US) 2005-05-31 US disclosed
EP-1532132-A1 NOVEL BENZODIOXOLES F.HOFFMANN-LA ROCHE AG (CH) 2005-05-25 EP disclosed
US-20040142922-A1 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. 2004-07-22 US disclosed
WO-2004013120-A1 NOVEL BENZODIOXOLES F. HOFFMANN-LA ROCHE AG (CH) 2004-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143373-A1 Benzodioxole derivatives CNR2, CNR1, GPR119 ALDH1A1 607/4885TSHR 1029/4885KIF11 4299/4885
US-20040142922-A1 Benzodioxole derivatives CNR1, CNR2, GPR119 ALDH1A1 299/4885TSHR 1171/4885KIF11 4326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.