SCHEMBL6076169

SCHEMBL6076169

CCCCc1cc(Cl)c2nc(C)c(C)c(OC(C)=O)c2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.34
EIF4A1 P60842 2/20 0.34
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
CTRC Q99895 1/20 0.33
HTT P42858 2/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 1/20 0.32
NR4A2 P43354 1/20 0.32
PTGES O14684 1/20 0.31
KDM4E B2RXH2 1/20 0.31
OPRM1 P35372 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
CNR2 P34972 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6077824 0.88 ALOX5 (0.36) ALOX5HTTNPC1HPGDMAPK1
SCHEMBL6076307 0.87 EIF4A1 (0.35) ALOX5EIF4A1HTTNPC1HPGD
SCHEMBL6077311 0.86 ALOX5 (0.36) ALOX5HTTNPC1HPGDMAPK1
SCHEMBL6078666 0.85 ALOX5 (0.36) ALOX5HTTNPC1HPGDMAPK1
SCHEMBL6077713 0.85 ALOX5 (0.44) ALOX5HPGDMAPK1LMNAKDM4E
SCHEMBL6076793 0.85 ALOX5 (0.40) ALOX5HTTHPGDLMNAKDM4E
SCHEMBL6076615 0.84 ALOX5 (0.33) ALOX5HTTNPC1HPGDMAPK1
SCHEMBL6076165 0.77 DHODH (0.32) HTTMAPK1NPSR1LMNAKDM4E
SCHEMBL6077005 0.75 DHODH (0.43) ALOX5LMNAALDH1A1
SCHEMBL845559 0.71 HTT (0.46) ALOX5HTTNPC1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067668-B2 4-quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture MEIJI SEIKA KAISHA, LTD. (JP) 2006-06-27 US disclosed
EP-0990648-B1 4-QUINOLINOL DERIVATIVES AND AGROHORTICULTURAL BACTERICIDES CONTAINING THE SAME AS ACTIVE INGREDIENT MEIJI SEIKA KAISHA (JP) 2005-11-02 EP disclosed
US-20040152728-A1 4-Quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture MEIJI SEIKA KAISHA, LTD. (JP) 2004-08-05 US disclosed
US-6680282-B2 FUNGICIDE HAVING AN EXCELLENT CONTROL EFFECT; 4-QUINOLINOL DERIVATIVES HAVING SPECIFIC SUBSTITUENT AT 1,2 AND ATLEAST ONE SUBSTITUENT AT 5,6,7,8 POSITION MEIJI SEIKA KAISHA, LTD. (JP) 2004-01-20 US disclosed
US-20030119863-A1 4-Quinolinol derivatives and agrohorticultural bactericides containing the same as active ingredient MEIJI SEIKA PHARMA CO., LTD. (JP) 2003-06-26 US disclosed
EP-0990648-A1 4-QUINOLINOL DERIVATIVES AND AGROHORTICULTURAL BACTERICIDES CONTAINING THE SAME AS ACTIVE INGREDIENT Meiji Seika Kaisha, Ltd. (JP) 2000-04-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040152728-A1 4-Quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture CYP51A1, CYP4X1, CYP4Z1 ALOX5 2069/4885EIF4A1 1012/4885AKR1C2 532/4885
US-20030119863-A1 4-Quinolinol derivatives and agrohorticultural bactericides containing the same as active ingredient CYP51A1, DDT, PGLS ALOX5 2036/4885EIF4A1 1618/4885AKR1C2 1008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.