Tyrphostin Ag 879

Tyrphostin Ag 879

SCHEMBL607701

CC(C)(C)c1cc(/C=C(\C#N)C(N)=S)cc(C(C)(C)C)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 1.00
KMT2A Q03164 8/20 1.00
ALDH1A1 P00352 8/20 1.00
MEN1 O00255 7/20 1.00
BLM P54132 6/20 1.00
HPGD P15428 6/20 1.00
TDP1 Q9NUW8 6/20 1.00
KDM4E B2RXH2 5/20 1.00
CYP3A4 P08684 4/20 1.00
TSHR P16473 4/20 1.00
HSD17B10 Q99714 4/20 1.00
RECQL P46063 4/20 1.00
ERBB2 P04626 3/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
RGS12 O14924 3/20 1.00
CYP1A2 P05177 3/20 1.00
CYP2C9 P11712 3/20 1.00
ALOX15 P16050 3/20 1.00
NFKB1 P19838 3/20 1.00
CYP2C19 P33261 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tyrphostin Ag 879 SCHEMBL607702 1.00 MAPT (1.00) MAPTKMT2AALDH1A1MEN1BLM
Tyrphostin Ag 879 SCHEMBL607703 1.00 MAPT (1.00) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL25736022 0.88 MEN1 (0.78) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL11093690 0.86 EGFR (1.00) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL20333049 0.86 MEN1 (0.76) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL11093692 0.86 EGFR (1.00) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL8346188 0.81 EGFR (0.76) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL6286531 0.81 MAPT (0.68) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL6278934 0.81 MAPT (0.68) MAPTKMT2AALDH1A1MEN1BLM
SCHEMBL3244723 0.80 EGFR (0.74) MAPTKMT2AALDH1A1MEN1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 947 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4709874-A1 MODULATORS OF PROTEIN SECRETION Sanofi (FR) 2026-03-18 EP claimed
US-20250129429-A1 GENE FUSIONS IN SARCOMA FOUNDATION MEDICINE, INC. (US) 2025-04-24 US claimed
WO-2024231896-A1 MODULATORS OF PROTEIN SECRETION SANOFI (FR) 2024-11-14 WO claimed
EP-4423302-A2 NOVEL KINASE FUSIONS DETECTED BY LIQUID BIOPSY Foundation Medicine, Inc. (US) 2024-09-04 EP claimed
US-20240287616-A1 METHODS OF DETECTING NTRK FUSION PROTEINS STRATA ONCOLOGY INC (US) 2024-08-29 US claimed
CN-118414439-A Novel kinase fusion by liquid biopsy 基金会医学公司 2024-07-30 CN claimed
EP-4399330-A1 GENE FUSIONS IN SARCOMA Foundation Medicine, Inc. (US) 2024-07-17 EP claimed
US-20240218051-A1 MODIFIED BINDING POLYPEPTIDES FOR OPTIMIZED DRUG CONJUGATION GENZYME CORPORATION 2024-07-04 US claimed
EP-3303610-B1 COMPOSITIONS AND METHODS FOR SCREENING SOLID TUMORS QUEST DIAGNOSTICS INVEST INC (US) 2024-05-08 EP claimed
EP-4355917-A1 METHODS OF DETECTING NTRK FUSION PROTEINS Strata Oncology, Inc. (US) 2024-04-24 EP claimed
EP-4126234-A1 COMPOSITIONS FOR CORONAVIRUS INFECTION TREATMENT AND/OR PREVENTION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-02-08 EP claimed
EP-4110404-A1 MODIFIED BINDING POLYPEPTIDES FOR OPTIMIZED DRUG CONJUGATION GENZYME CORPORATION (US) 2023-01-04 EP claimed
CN-115515643-A Modified binding polypeptides for optimized drug conjugation 建新公司 2022-12-23 CN claimed
WO-2022266551-A1 METHODS OF DETECTING NTRK FUSION PROTEINS Strata Oncology, Inc. (US) 2022-12-22 WO claimed
US-11525008-B2 Methods and pharmaceutical compositions for the treatment of lung cancer INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2022-12-13 US claimed
CN-115474430-A Composition for treatment and/or prevention of coronavirus infection 弗劳恩霍夫应用研究促进协会 2022-12-13 CN claimed
US-20220243280-A1 NTRK FUSION MOLECULES AND USES THEREOF FOUNDATION MEDICINE, INC. (US) 2022-08-04 US claimed
EP-3980563-A2 NTRK FUSION MOLECULES AND USES THEREOF Foundation Medicine, Inc. (US) 2022-04-13 EP claimed
US-6596878-B2 Protein kinase inhibitor compositio; used to treat cell proliferative disorders such as cancers charcterized by over-activity or inappropriate activity HER2 or EGFR. YISSUM RESEARCH & DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY (IL) 2003-07-22 US claimed
US-5981569-A CAPABLE OF MODULATING TYROSINE KINASE SIGNAL TRANSDUCTION AND PARTICULARLY KDR/FLK-1 RECEPTOR SIGNAL TRANSDUCTION IN ORDER TO REGULATE AND/OR MODULATE VASCULOGENESIS AND ANGIOGENESIS; TREATMENT OF CANCER, DIABETES, HEMANGIOMA YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1999-11-09 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220243280-A1 NTRK FUSION MOLECULES AND USES THEREOF NTRK1, NTRK3, NTRK2 MAPT 2245/4885KMT2A 4235/4885ALDH1A1 4003/4885
US-11525008-B2 Methods and pharmaceutical compositions for the treatment of lung cancer FHIT, MAT2A, MAT1A MAPT 4334/4885KMT2A 289/4885ALDH1A1 1045/4885
US-20240218051-A1 MODIFIED BINDING POLYPEPTIDES FOR OPTIMIZED DRUG CONJUGATION FCGR3B, CD2BP2, FCGR2A MAPT 1888/4885KMT2A 3604/4885ALDH1A1 2301/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.