SCHEMBL6077221

SCHEMBL6077221

O=C(O)C1=C(O)C(=O)N(CCN2CCN(C(Cc3ccccc3)C3=COCO3)CC2)C1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 7/20 0.35
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 1/20 0.30
PARP1 P09874 1/20 0.30
ACHE P22303 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15961230 0.75 SIGMAR1 (0.52) CYP1A2CYP2D6TSHRCYP2C19ALDH1A1
SCHEMBL2853081 0.75 CHRM1 (0.41) CYP1A2CYP3A4CYP2D6TSHRCYP2C19
SCHEMBL2316904 0.74 SIGMAR1 (0.47) CYP1A2CYP3A4CYP2D6TSHRCYP2C19
SCHEMBL2116312 0.72 ADRB1 (0.48)
SCHEMBL3708454 0.71 CYP1A2 (0.40) CYP1A2CYP3A4CYP2D6TSHRCYP2C19
SCHEMBL3591699 0.70 FAAH (0.50) TSHRCYP2C19
SCHEMBL6076770 0.69 KMT2A (0.53) TSHRALDH1A1
Hydrochloric Acid SCHEMBL3605151 0.69 FAAH (0.49) TSHRCYP2C19
SCHEMBL592971 0.69 SLC6A4 (0.61) CYP1A2CYP2D6CYP2C19
SCHEMBL217536 0.69 CYP1A2 (0.42) CYP1A2CYP3A4CYP2D6TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109186-B2 4-hydroxy-5-oxo-1-(2-[4-methylpiperazin-1-yl]ethyl)-2,5-dihydro-1H-pyrrole-3-carboxylic acid (3,4-dichlorobenzyl)-methyl-amide for human immunodeficiency virus (HIV) treatment BRISTOL-MYERS SQUIBB COMPANY (US) 2006-09-19 US disclosed
US-20040110804-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040110804-A1 HIV integrase inhibitors CDKN1A, SAMHD1, CTCF LIPG 2895/4885CYP1A2 483/4885CYP3A4 461/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.