SCHEMBL6081708

SCHEMBL6081708

O=C1NC(=O)c2c1c1c3cc(OCc4ccccc4)ccc3[nH]c1c1cccn21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.61
CDK4 P11802 2/20 0.51
CCND1 P24385 2/20 0.51
CCNE2 O96020 1/20 0.51
PRKACA P17612 1/20 0.51
PRKACG P22612 1/20 0.51
PRKACB P22694 1/20 0.51
CCNE1 P24864 1/20 0.51
CDK2 P24941 1/20 0.51
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
ROCK2 O75116 2/20 0.46
CTSV O60911 3/20 0.45
CTSL P07711 3/20 0.45
PDGFRB P09619 1/20 0.45
WEE1 P30291 2/20 0.44
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080842 0.86 CHEK1 (0.52) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL6081478 0.80 ROCK2 (0.64) CHEK1CDK4ROCK2WEE1
SCHEMBL6081058 0.79 CDK4 (0.50) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL6080997 0.78 CDK4 (0.61) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL6080935 0.78 CDK4 (0.60) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL9623279 0.74 CHEK1 (0.64) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL5879186 0.72 MAOA (0.58) CHEK1MAOAMAOBCTSVCTSL
SCHEMBL5879315 0.70 MAOB (0.54) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL6080498 0.69 CDK4 (0.56) CHEK1CDK4CCND1CCNE2PRKACA
SCHEMBL13711924 0.69 PARP1 (0.61) CHEK1MAOAMAOBCTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060004428-A1 Pyrrolo (3,4-c) carbazole and pyrido (2,3-b) pyrrolo (3,4-e) indole derivatives, preparation method and pharmaceutical compositions containing same LES LABORATOIRES SERVIER (FR) 2006-01-05 US disclosed