SCHEMBL6080498

SCHEMBL6080498

O=C1NC(=O)c2c1c1c3cccnc3[nH]c1c1cccn21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 8/20 0.56
CCND1 P24385 8/20 0.56
GSK3B P49841 4/20 0.41
CLK1 P49759 1/20 0.41
CHEK1 O14757 3/20 0.39
PARP1 P09874 2/20 0.38
AURKA O14965 1/20 0.38
FEN1 P39748 1/20 0.38
PRKCA P17252 2/20 0.38
CDK5 Q00535 2/20 0.38
CDK5R1 Q15078 2/20 0.38
MEN1 O00255 1/20 0.38
PRKD3 O94806 1/20 0.38
CCNB2 O95067 1/20 0.38
CCNE2 O96020 1/20 0.38
PRKCG P05129 1/20 0.38
PRKCB P05771 1/20 0.38
CDK1 P06493 1/20 0.38
MAPT P10636 1/20 0.38
CCNB1 P14635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080997 0.81 CDK4 (0.61) CDK4CCND1GSK3BCHEK1PARP1
SCHEMBL22566992 0.79 CDK4 (0.83) CDK4CCND1GSK3BCHEK1PARP1
SCHEMBL6081058 0.74 CDK4 (0.50) CDK4CCND1GSK3BCLK1CHEK1
SCHEMBL6081478 0.73 ROCK2 (0.64) CDK4GSK3BCLK1CHEK1PRKCA
SCHEMBL6080935 0.73 CDK4 (0.60) CDK4CCND1GSK3BCLK1CHEK1
SCHEMBL9262153 0.72 CDK4 (1.00) CDK4CCND1GSK3BCHEK1PARP1
SCHEMBL14346099 0.69 PARP1 (0.66) CDK4CCND1CHEK1PARP1
SCHEMBL6081708 0.69 CHEK1 (0.61) CDK4CCND1CHEK1CCNE2PRKACA
SCHEMBL9259173 0.68 CDK4 (0.74) CDK4CCND1GSK3BCHEK1PRKCA
SCHEMBL6081576 0.67 CDK4 (0.41) CDK4CCND1GSK3BCLK1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060004428-A1 Pyrrolo (3,4-c) carbazole and pyrido (2,3-b) pyrrolo (3,4-e) indole derivatives, preparation method and pharmaceutical compositions containing same LES LABORATOIRES SERVIER (FR) 2006-01-05 US disclosed